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Volume 189

European Journal of Medicinal Chemistry

Volume 189

1

Synthesis and SARs of dopamine derivatives as potential inhibitors of influenza virus PAN endonuclease

Liao, Yixian, Ye, Yilu, Li, Sumei, Zhuang, Yilian, Chen, Liye, Chen, Jianxin, Cui, Zining, Huo, Lijian, Liu, Shuwen, Song, Gaopeng

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.07 MB

2020

2

Discovery of potent epidermal growth factor receptor (EGFR) degraders by proteolysis targeting chimera (PROTAC)

Zhang, Hao, Zhao, Hong-Yi, Xi, Xiao-Xiao, Liu, Yan-Jie, Xin, Minhang, Mao, Shuai, Zhang, Jun-Jie, Lu, A-Xin, Zhang, San-Qi

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 8.00 MB

2020

3

β-Lactams with antiproliferative and antiapoptotic activity in breast and chemoresistant colon cancer cells

Malebari, Azizah M., Fayne, Darren, Nathwani, Seema M., O’Connell, Fiona, Noorani, Sara, Twamley, Brendan, O’Boyle, Niamh M., O’Sullivan, Jacintha, Zisterer, Daniela M., Meegan, Mary J.

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 2.51 MB

2020

4

Synthesis, biological evaluation and in silico modeling of novel integrase strand transfer inhibitors (INSTIs)

Ivashchenko, Andrey A., Ivanenkov, Yan A., Koryakova, Angela G., Karapetian, Ruben N., Mitkin, Oleg D., Aladinskiy, Vladimir A., Kravchenko, Dmitry V., Savchuk, Nikolai P., Ivashchenko, Alexander V.

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.45 MB

2020

5

Synthesis, mechanisms of action, and toxicity of novel aminophosphonates derivatives conjugated irinotecan in vitro and in vivo as potent antitumor agents

Huang, Xiaochao, Wang, Meng, You, Qinghong, Kong, Jing, Zhang, Haijiang, Yu, Chunhao, Wang, Yanming, Wang, Hengshan, Huang, Rizhen

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 671 KB

2020

6

Synthetic tumor-specific antigenic peptides with a strong affinity to HLA-A2 elicit anti-breast cancer immune response through activating CD8+ T cells

Shi, Wei, Qiu, Qianqian, Tong, Zhenzhen, Guo, Weiwei, Zou, Feng, Feng, Ziying, Wang, Yao, Huang, Wenlong, Qian, Hai

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Langue:

english

Fichier:

PDF, 3.71 MB

english, 2020

7

Simple amphiphilic α-hydrazido acids: Rational design, synthesis, and in vitro bioactivity profile of a novel class of potential antimicrobial compounds

Amabili, Paolo, Biavasco, Francesca, Brenciani, Andrea, Citterio, Barbara, Corbisiero, Dario, Ferrazzano, Lucia, Fioriti, Simona, Guerra, Giulia, Orena, Mario, Rinaldi, Samuele

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Langue:

english

Fichier:

PDF, 2.76 MB

english, 2020

8

Celastrol: Progresses in structure-modifications, structure-activity relationships, pharmacology and toxicology

Hou, Wei, Liu, Bo, Xu, Hongtao

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.18 MB

2020

9

Identification of descriptors for structure-activity relationship in ruthenium (II) mixed compounds with antiparasitic activity

Cedillo-GutiÃ©rrez, Erika Lorena, HernÃ¡ndez-Ayala, Luis Felipe, Torres-GutiÃ©rrez, Carolina, Reina, Miguel, Flores-Alamo, Marcos, Carrero, Julio C., Ugalde-SaldÃvar, VÃctor M., Ruiz-Azuara, Lena

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.40 MB

2020

10

Dammarane-type leads panaxadiol and protopanaxadiol for drug discovery: Biological activity and structural modification

Wang, Mingying, Li, Haonan, Liu, Weiwei, Cao, Hao, Hu, Xu, Gao, Xiang, Xu, Fanxing, Li, Zhanlin, Hua, Huiming, Li, Dahong

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Langue:

english

Fichier:

PDF, 3.72 MB

english, 2020

11

Optimization of EphA2 antagonists based on a lithocholic acid core led to the identification of UniPR505, a new 3Î±-carbamoyloxy derivative with antiangiogenetic properties

Incerti, Matteo, Russo, Simonetta, Corrado, Miriam, Giorgio, Carmine, Ballabeni, Vigilio, Chiodelli, Paola, Rusnati, Marco, Scalvini, Laura, Callegari, Donatella, Castelli, Riccardo, Vacondio, Federic

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Langue:

english

Fichier:

PDF, 2.81 MB

english, 2020

12

Graphical abstract TOC continued

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 3.34 MB

2020

13

Editorial Board

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 47 KB

2020

14

Graphical abstract TOC

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 359 KB

2020

15

Graphical abstract TOC

Journal:

European Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 275 KB

2020