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Volume 163

European Journal of Medicinal Chemistry

Volume 163

1

Discovery of novel anti-angiogenesis agents. Part 10: Multi-target inhibitors of VEGFR-2, Tie-2 and EphB4 incorporated with 1,2,3-triazol

Pan, Xiaoyan, Liang, Liyuan, Si, Ru, Wang, Jin, Zhang, Qingqing, Zhou, Huaxin, Zhang, Lin, Zhang, Jie

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 1.60 MB

english, 2019

2

Tailoring a lead-like compound targeting multiple G-quadruplex structures

Amato, Jussara, Platella, Chiara, Iachettini, Sara, Zizza, Pasquale, Musumeci, Domenica, Cosconati, Sandro, Pagano, Alessia, Novellino, Ettore, Biroccio, Annamaria, Randazzo, Antonio, Pagano, Bruno, M

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 2.99 MB

english, 2019

3

Chemistry-oriented synthesis (ChOS) and target deconvolution on neuroprotective effect of a novel scaffold, oxaza spiroquinone

Venkanna, Arramshetti, Cho, Kyo Hee, Dhorma, Lama Prema, Kumar, Duddukuri Nandan, Hah, Jung Mi, Park, Hyeung-geun, Kim, Sun Yeou, Kim, Mi-hyun

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 4.05 MB

english, 2019

4

In vitro and in vivo anti-tumor activity of two gold(III) complexes with isoquinoline derivatives as ligands

Khan, Taj-Malook, Gul, Noor Shad, Lu, Xing, Wei, Jian-Hua, Liu, Yan-Cheng, Sun, Hongbin, Liang, Hong, Orvig, Chris, Chen, Zhen-Feng

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 3.21 MB

english, 2019

5

Exploring structural properties of potent human carbonic anhydrase inhibitors bearing a 4-(cycloalkylamino-1-carbonyl)benzenesulfonamide moiety

Buemi, Maria Rosa, Di Fiore, Anna, De Luca, Laura, Angeli, Andrea, Mancuso, Francesca, Ferro, Stefania, Monti, Simona Maria, Buonanno, Martina, Russo, Emilio, De Sarro, Giovanbattista, De Simone, Gius

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 1.90 MB

english, 2019

6

Polycyclic maleimide-based derivatives as first dual modulators of neuronal calcium channels and GSK-3β for Alzheimer's disease treatment

Bisi, Alessandra, Arribas, Raquel L., Micucci, Matteo, Budriesi, Roberta, Feoli, Alessandra, Castellano, Sabrina, Belluti, Federica, Gobbi, Silvia, de los Rios, Cristobal, Rampa, Angela

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 1.10 MB

english, 2019

7

Fragment-based drug discovery of triazole inhibitors to block PDEδ-RAS protein-protein interaction

Chen, Danqi, Chen, Yuehong, Lian, Fulin, Chen, Liu, Li, Yanlian, Cao, Danyan, Wang, Xin, Chen, Lin, Li, Jian, Meng, Tao, Huang, Min, Geng, Meiyu, Shen, Jingkang, Zhang, Naixia, Xiong, Bing

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 1.61 MB

english, 2019

8

Synthesis and anti-tumor activity of imidazopyrazines as TAK1 inhibitors

Kang, Seok Jong, Lee, Jung Wuk, Chung, Shin Hyuck, Jang, Sun Young, Choi, Jaeyul, Suh, Kwee Hyun, Kim, Young Hoon, Ham, Young Jin, Min, Kyung Hoon

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 750 KB

english, 2019

9

The p53 stabilizing agent CP-31398 and multi-kinase inhibitors. Designing, synthesizing and screening of styrylquinazoline series

Mularski, Jacek, Malarz, Katarzyna, Pacholczyk, Marcin, Musiol, Robert

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 1.82 MB

english, 2019

10

Design, synthesis, and evaluation of fluorine and Naphthyridine–Based half-sandwich organoiridium/ruthenium complexes with bioimaging and anticancer activity

Li, JuanJuan, Tian, Zhenzhen, Ge, Xingxing, Xu, Zhishan, Feng, Yaqian, Liu, Zhe

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 2.11 MB

english, 2019

11

Discovery of novel quaternary ammonium compounds based on quinuclidine-3-ol as new potential antimicrobial candidates

Bazina, Linda, Maravić, Ana, Krce, Lucija, Soldo, Barbara, Odžak, Renata, Popović, Viljemka Bučević, Aviani, Ivica, Primožič, Ines, Šprung, Matilda

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 1.33 MB

english, 2019

12

Discovery, synthesis and anti-atherosclerotic activities of a novel selective sphingomyelin synthase 2 inhibitor

Li, Yali, Huang, Taomin, Lou, Bin, Ye, Deyong, Qi, Xiangyu, Li, Xiaoxia, Hu, Shuang, Ding, Tingbo, Chen, Yan, Cao, Yang, Mo, Mingguang, Dong, Jibin, Wei, Min, Chu, Yong, Li, Huiti, Jiang, Xian-Cheng,

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 1.67 MB

english, 2019

13

Discovery and optimization of a series of 3-substituted indazole derivatives as multi-target kinase inhibitors for the treatment of lung squamous cell carcinoma

Wang, Qi, Dai, Yang, Ji, Yinchun, Shi, Huanyu, Guo, Zuhao, Chen, Danqi, Chen, Yuelei, Peng, Xia, Gao, Yinglei, Wang, Xin, Chen, Lin, Jiang, Yuchen, Geng, Meiyu, Shen, Jingkang, Ai, Jing, Xiong, Bing

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 3.44 MB

english, 2019

14

Discovery of novel nonsteroidal VDR agonists with novel diarylmethane skeleton for the treatment of breast cancer

Wang, Cong, Wang, Bin, Hou, Siyuan, Xue, Lingjing, Kang, Zisheng, Du, Junjie, Li, Yanyi, Liu, Xuwentai, Wang, Qianqian, Zhang, Can

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 3.11 MB

english, 2019

15

Corrigendum to ‘Synthesis and discovery of a drug candidate for treatment of idiopathic pulmonary fibrosis through inhibition of TGF-b1 pathway’ [Eur. J. Med. Chem. 157 (2018) 229–247]

Li, Xiaohe, Lu, Cheng, Liu, Shuangwei, Liu, Shuaishuai, Su, Chengcheng, Xiao, Ting, Bi, Zhun, Sheng, Pengzhen, Huang, Mengying, Liu, Xinhua, Wei, Yujiao, Zhao, Lin, Miao, Shengxiang, Mao, Jiahe, Huang

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Langue:

english

Fichier:

PDF, 172 KB

english, 2019

16

Editorial Board

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Fichier:

PDF, 410 KB

2019

17

Graphical abstract TOC

Journal:

European Journal of Medicinal Chemistry

Année:

2019

Fichier:

PDF, 275 KB

2019