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Volume 150

European Journal of Medicinal Chemistry

Volume 150

1

Evaluation of the novel TSPO radiotracer 2-(7-butyl-2-(4-(2-([ 18 F]fluoroethoxy)phenyl)-5-methylpyrazolo[1,5- a ]pyrimidin-3-yl)- N , N -diethylacetamide in a preclinical model of neuroinflammation

Tang, Dewei, Fujinaga, Masayuki, Hatori, Akiko, Zhang, Yiding, Yamasaki, Tomoteru, Xie, Lin, Mori, Wakana, Kumata, Katsushi, Liu, Jianjun, Manning, H. Charles, Huang, Gang, Zhang, Ming-Rong

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 1.14 MB

english, 2018

2

The aminopyridine-3,5-dicarbonitrile core for the design of new non-nucleoside-like agonists of the human adenosine A 2B receptor

Betti, Marco, Catarzi, Daniela, Varano, Flavia, Falsini, Matteo, Varani, Katia, Vincenzi, Fabrizio, Ben, Diego Dal, Lambertucci, Catia, Colotta, Vittoria

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 1.92 MB

english, 2018

3

Anti-inflammatory hybrids of secondary amines and amide-sulfamide derivatives

Bai, Renren, Sun, Jian, Liang, Zhongxing, Yoon, Younghyoun, Salgado, Eric, Feng, Amber, Oum, Yoonhyeun, Xie, Yuanyuan, Shim, Hyunsuk

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 2.71 MB

english, 2018

4

Polypharmacology in HIV inhibition: can a drug with simultaneous action against two relevant targets be an alternative to combination therapy?

de Castro, Sonia, Camarasa, María-José

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 2.16 MB

english, 2018

5

Discovery of 4-(( N -(2-(dimethylamino)ethyl)acrylamido)methyl)- N -(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFRα kinase inhibitor for PDGFRα driving chronic eosinophilic leukemia

Wang, Qiang, Liu, Feiyang, Qi, Shuang, Qi, Ziping, Yan, Xiao-E., Wang, Beilei, Wang, Aoli, Wang, Wei, Chen, Cheng, Liu, Xiaochuan, Jiang, Zongru, Hu, Zhenquan, Wang, Li, Wang, Wenchao, Ren, Tao, Zhang

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 4.99 MB

english, 2018

6

Design, synthesis, biological evaluation and in vivo testing of dual phosphodiesterase 5 (PDE5) and histone deacetylase 6 (HDAC6)-selective inhibitors for the treatment of Alzheimer's disease

Rabal, Obdulia, Sánchez-Arias, Juan A., Cuadrado-Tejedor, Mar, de Miguel, Irene, Pérez-González, Marta, García-Barroso, Carolina, Ugarte, Ana, Estella-Hermoso de Mendoza, Ander, Sáez, Elena, Espelosin

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 1.69 MB

english, 2018

7

Synthesis and biological evaluation of nannocystin analogues toward understanding the binding role of the (2 R ,3 S )-Epoxide in nannocystin A

Tian, Yunfeng, Xu, Xiaolong, Ding, Yahui, Hao, Xin, Bai, Yanju, Tang, Yang, Zhang, Xuemei, Li, Qiuying, Yang, Zhantao, Zhang, Weicheng, Chen, Yue

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 1.26 MB

english, 2018

8

1-Aroylindoline-hydroxamic acids as anticancer agents, inhibitors of HSP90 and HDAC

Ojha, Ritu, Huang, Han-Li, HuangFu, Wei-Chun, Wu, Yi-Wen, Nepali, Kunal, Lai, Mei-Jung, Su, Chih-Jou, Sung, Ting-Yi, Chen, Yi-Lin, Pan, Shiow-Lin, Liou, Jing-Ping

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 1.02 MB

english, 2018

9

Synthesis of 3′-halo-5′-norcarbocyclic nucleoside phosphonates as potent anti-HIV agents

Hamon, Nadège, Kaci, Malika, Uttaro, Jean-Pierre, Périgaud, Christian, Mathé, Christophe

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 1.18 MB

english, 2018

10

N,N′ -disubstituted cinnamamide derivatives potentiate ciprofloxacin activity against overexpressing NorA efflux pump Staphylococcus aureus 1199B strains

Radix, Sylvie, Jordheim, Anne Doléans, Rocheblave, Luc, N'Digo, Serge, Prignon, Anne-Laure, Commun, Carine, Michalet, Serge, Dijoux-Franca, Marie-Geneviève, Mularoni, Angélique, Walchshofer, Nadia

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 596 KB

english, 2018

11

Editorial Board

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Fichier:

PDF, 206 KB

2018

12

Graphical abstract TOC

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Fichier:

PDF, 293 KB

2018

13

Graphical abstract TOC

Journal:

European Journal of Medicinal Chemistry

Année:

2018

Fichier:

PDF, 443 KB

2018