Volume 80; Issue 4

Chemical Biology & Drug Design

Volume 80; Issue 4

1

Anticonvulsant Activity of Novel 1-(Substituted Benzylidene)-4-(1-(Morpholino/Piperidino Methyl)-2,3-Dioxoindolin-5-yl) Semicarbazide Derivatives in Mice and Rats Acute Seizure Models

Chinnasamy Rajaram Prakash, Sundararajan Raja, Govindaraj Saravanan

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 152 KB

english, 2012

2

Novel Benzimidazole Analogs as Inhibitors of EGFR Tyrosine Kinase

Soni Yadav, Deepa Sinha, Sanjay K. Singh, Vinay K. Singh

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 212 KB

english, 2012

3

Ligand- and Structure-Based Drug Design Strategies and PPARδ/α Selectivity

Vinícius G. Maltarollo, Káthia M. Honório

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 879 KB

english, 2012

4

Complexes of an Alpha Thymosin Derivative with 185/187Re and 99mTc: Structural Analysis and Initial Biological Evaluation

Dimitra Benaki, Christos Zikos, Chrysoula-Evangelia Karachaliou, Ourania Tsitsilonis, Leondios Leondiadis, Hubert Kalbacher, Wolfgang Voelter, Minas Papadopoulos, Ioannis Pirmettis, Maria Pelecanou, E

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 283 KB

english, 2012

5

An Isoquinoline Alkaloid, Berberine, Can Inhibit Fungal Alpha Amylase: Enzyme Kinetic and Molecular Modeling Studies

Ignatius Tintu, Kalarickal V Dileep, Anu Augustine, Chittalakkottu Sadasivan

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 317 KB

english, 2012

6

Identification of FDA-approved Drugs that Computationally Bind to MDM2

Wayne A. Warner, Ricardo Sanchez, Alex Dawoodian, Esther Li, Jamil Momand

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 383 KB

english, 2012

7

Molecular Dynamics Simulations of Peptide Inhibitors Complexed With Trypanosoma cruzi Trypanothione Reductase

Samuel Silva Da Rocha Pita, Paulo Ricardo Batista, Magaly Girão Albuquerque, Pedro Geraldo Pascutti

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 515 KB

english, 2012

8

Design, Synthesis, Antibacterial Activity, and Molecular Docking Studies of Novel Hybrid 1,3-Thiazine-1,3,5-Triazine Derivatives as Potential Bacterial Translation Inhibitor

Udaya P. Singh, Manish Pathak, Vaibhav Dubey, Hans R. Bhat, Prashant Gahtori, Ramendra K. Singh

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 286 KB

english, 2012

9

Synthesis and Biological Evaluation of 2,4,6-Trihydroxychalcone Derivatives as Novel Protein Tyrosine Phosphatase 1B Inhibitors

Liang-Peng Sun, Li-Xin Gao, Wei-Ping Ma, Fa-Jun Nan, Jia Li, Hu-Ri Piao

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 287 KB

english, 2012

10

Replacement of the Methylene of Dihydrochalcones with Oxygen: Synthesis and Biological Evaluation of 2-Phenoxyacetophenones

Mahsa Ansari, Saeed Emami, Mohammad A. Khalilzadeh, Malek T. Maghsoodlou, Alireza Foroumadi, Mohammad A. Faramarzi, Nasrin Samadi, Sussan K. Ardestani

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 151 KB

english, 2012

11

Design, Facile Synthesis, and Antibacterial Activity of Hybrid 1,3,4-thiadiazole-1,3,5-triazine Derivatives Tethered via –S– Bridge

Vaibhav Dubey, Manish Pathak, Hans R. Bhat, Udaya P. Singh

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 177 KB

english, 2012

12

Synthesis and Biological Evaluation of 3-thiazolocoumarinyl Schiff-base Derivatives as Cholinesterase Inhibitors

Rabia Raza, Aamer Saeed, Mubeen Arif, Shamsul Mahmood, Muhammad Muddassar, Ahsan Raza, Jamshed Iqbal

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 600 KB

english, 2012

13

Design, Synthesis, and Evaluation of 2-(arylsulfonyl)oxiranes as Cell-permeable Covalent Inhibitors of Protein Tyrosine Phosphatases

Dibyendu Dana, Tirtha K. Das, Ish Kumar, Anibal R. Davalos, Kevin J. Mark, Daryl Ramai, Emmanuel J. Chang, Tanaji T. Talele, Sanjai Kumar

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 269 KB

english, 2012

14

Neoflavonoids and Tetrahydroquinolones as Possible Cancer Chemopreventive Agents

Suaib Luqman, Abha Meena, Pragya Singh, Tamara P. Kondratyuk, Laura E. Marler, John M. Pezzuto, Arvind S. Negi

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 668 KB

english, 2012

15

Synthesis and Kinetic Testing of Tetrahydropyrimidine-2-thione and Pyrrole Derivatives as Inhibitors of the Metallo-β-lactamase from Klebsiella pneumonia and Pseudomonas aeruginosa

Waleed M. Hussein, Samar S. Fatahala, Zainab M. Mohamed, Ross P. McGeary, Gerhard Schenk, David L. Ollis, Mosaad S. Mohamed

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 1.73 MB

english, 2012

16

Click Chemistry Approach for Bis-Chromenyl Triazole Hybrids and Their Antitubercular Activity

Reshma J. Naik, Manohar V. Kulkarni, K. Sreedhara Ranganath Pai, Pawan G. Nayak

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 180 KB

english, 2012

17

Issue Information

Journal:

Chemical Biology & Drug Design

Année:

2012

Langue:

english

Fichier:

PDF, 520 KB

english, 2012