Volume 28; Issue 24

Bioorganic & Medicinal Chemistry

Volume 28; Issue 24

1

Synthesis and biological evaluation of NQO1-activated prodrugs of podophyllotoxin as antitumor agents

Qu, Yan, Zhang, Chong, Ma, Xin, Gao, Yunhui, Liu, Jing, Wu, Liqiang

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 3.75 MB

2020

2

Identification of novel STAT3 inhibitors bearing 2-acetyl-7-phenylamino benzofuran scaffold for antitumour study

Wang, Feng, Feng, Kai-Rui, Zhao, Jia-Ying, Zhang, Jian-Wei, Shi, Xin-Wei, Zhou, Jian, Gao, Dingding, Lin, Guo-Qiang, Tian, Ping

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.75 MB

2020

3

One-step partial synthesis of (Â±)-asperteretone B and related hPTP1B1â400 inhibitors from butyrolactone I

Rivera-ChÃ¡vez, JosÃ©, Coporo-Blancas, Diego, Morales-JimÃ©nez, JesÃºs

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 2.55 MB

2020

4

Therapeutic strategies targeting somatic stem cells: Chemical approaches

Yu, Chen, Ding, Sheng

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 983 KB

2020

5

Bivalent HIV-1 fusion inhibitors based on peptidomimetics

Kobayakawa, Takuya, Ebihara, Kento, Tsuji, Kohei, Kawada, Takuma, Fujino, Masayuki, Honda, Yuzuna, Ohashi, Nami, Murakami, Tsutomu, Tamamura, Hirokazu

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.03 MB

2020

6

A dual-adjuvanting strategy for peptide-based subunit vaccines against group A Streptococcus: Lipidation and polyelectrolyte complexes

Zhao, Lili, Yang, Jieru, Nahar, Ummey Jannatun, Khalil, Zeinab G., Capon, Robert J., Hussein, Waleed M., Skwarczynski, Mariusz, Toth, Istvan

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.42 MB

2020

7

Special issue preface

Schultz, Peter G.

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 189 KB

2020

8

Antimalarial and anti-inflammatory activities of new chloroquine and primaquine hybrids: Targeting the blockade of malaria parasite transmission

Boechat, Nubia, Carvalho, Rita C.C., Ferreira, Maria de Lourdes G., Coutinho, Julia Penna, Sa, Paula M., Seito, Leonardo N., Rosas, Elaine C., Krettli, Antoniana U., Bastos, Monica M., Pinheiro, Luiz

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.00 MB

2020

9

Discovery of polypodiside as a Keap1-dependent Nrf2 activator attenuating oxidative stress and accumulation of extracellular matrix in glomerular mesangial cells under high glucose

Yao, Huankai, Zhang, Nan, Zhang, Wenting, Li, Jindong, Hua, Huilian, Li, Yan

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 5.55 MB

2020

10

Redirecting cytotoxic T cells with chemically programmed antibodies

Qi, Junpeng, Rader, Christoph

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.06 MB

2020

11

Discovery of a potent dual inhibitor of wild-type and mutant respiratory syncytial virus fusion proteins through the modulation of atropisomer interconversion properties

Yamaguchi-Sasaki, Toru, Kawaguchi, Takanori, Okada, Atsushi, Tokura, Seiken, Tanaka-Yamamoto, Nozomi, Takeuchi, Tomoki, Ogata, Yuya, Takahashi, Ryo, Kurimoto-Tsuruta, Risa, Tamaoki, Tomokazu, Sugaya,

Journal:

Bioorganic & Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.91 MB

2020