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Volume 14; Issue 5

Bioorganic & Medicinal Chemistry

Volume 14; Issue 5

1

Design, synthesis, and evaluation of novel galloyl pyrrolidine derivatives as potential anti-tumor agents

Xun Li, Yalin Li, Wenfang Xu

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 294 KB

english, 2006

2

Synthesis and in vitro activities of ferrocenic aminohydroxynaphthoquinones against Toxoplasma gondii and Plasmodium falciparum

Apiwat Baramee, Alexandra Coppin, Marlène Mortuaire, Lydie Pelinski, Stanislas Tomavo, Jacques Brocard

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 187 KB

english, 2006

3

Design, synthesis, and biological activity of novel factor Xa inhibitors: Improving metabolic stability by S1 and S4 ligand modification

Satoshi Komoriya, Shozo Kobayashi, Ken Osanai, Toshiharu Yoshino, Tsutomu Nagata, Noriyasu Haginoya, Yumi Nakamoto, Akiyoshi Mochizuki, Takayasu Nagahara, Makoto Suzuki, Takashi Shimada, Kengo Watanab

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 515 KB

english, 2006

4

Microwave enhanced solid support synthesis of fluorine containing benzopyrano-triazolo-thiadiazepines as potent anti-fungal agents

Anshu Dandia, Ruby Singh, Sarita Khaturia

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 140 KB

english, 2006

5

Affinity prediction on A1 adenosine receptor agonists: The chemometric approach

Paola Fossa, Luisa Mosti, Francesco Bondavalli, Silvia Schenone, Angelo Ranise, Chiara Casolino, Michele Forina

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 425 KB

english, 2006

6

Structure–intrinsic activity relationship studies in the group of 1-imido/amido substituted 4-(4-arylpiperazin-1-yl)cyclohexane derivatives; new, potent 5-HT1A receptor agents with anxiolytic- like activity

Andrzej J. Bojarski, Maria H. Paluchowska, Beata Duszyńska, Ryszard Bugno, Aleksandra Kłodzińska, Ewa Tatarczyńska, Ewa Chojnacka-Wójcik

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 236 KB

english, 2006

7

Discovery of potent and selective PARP-1 and PARP-2 inhibitors: SBDD analysis via a combination of X-ray structural study and homology modeling

Junya Ishida, Hirofumi Yamamoto, Yoshiyuki Kido, Kazunori Kamijo, Kenji Murano, Hiroshi Miyake, Mitsuru Ohkubo, Takayoshi Kinoshita, Masaichi Warizaya, Akinori Iwashita, Kayoko Mihara, Nobuya Matsuoka

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 576 KB

english, 2006

8

Synthesis of hypermodified adenosine derivatives as selective adenosine A3 receptor ligands

Liesbet Cosyn, Zhan-Guo Gao, Philippe Van Rompaey, Changrui Lu, Kenneth A. Jacobson, Serge Van Calenbergh

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 238 KB

english, 2006

9

Synthesis and biological evaluation of new non-imidazole H3-receptor antagonists of the 2-aminobenzimidazole series

Mirko Rivara, Valentina Zuliani, Giuseppe Cocconcelli, Giovanni Morini, Mara Comini, Silvia Rivara, Marco Mor, Fabrizio Bordi, Elisabetta Barocelli, Vigilio Ballabeni, Simona Bertoni, Pier Vincenzo Pl

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 275 KB

english, 2006

10

The 3D-QSAR analysis of 4(3H)-quinazolinone derivatives with dithiocarbamate side chains on thymidylate synthase

Shiying Liu, Feng Liu, Xiaoqing Yu, Guoyu Ding, Ping Xu, Jian Cao, Yuyang Jiang

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 517 KB

english, 2006

11

Inactivation of bovine plasma amine oxidase by haloallylamines

Jisook Kim, Yuming Zhang, Chongzhao Ran, Lawrence M. Sayre

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 266 KB

english, 2006

12

Human serum albumin interaction with formononetin studied using fluorescence anisotropy, FT-IR spectroscopy, and molecular modeling methods

Ying Li, WenYing He, YuMing Dong, Fenling Sheng, ZhiDe Hu

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 337 KB

english, 2006

13

New substrates and inhibitors of γ-aminobutyric acid aminotransferase containing bioisosteres of the carboxylic acid group: Design, synthesis, and biological activity

Hai Yuan, Richard B. Silverman

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 190 KB

english, 2006

14

Stereoselective synthesis and anti-inflammatory activities of 6- and 7-membered dioxacycloalkanes

Keli Gu, Lanrong Bi, Ming Zhao, Chao Wang, Cheryl Dolan, Michael C. Kao, Jeffrey B.-H. Tok, Shiqi Peng

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 175 KB

english, 2006

15

Structural basis for DNA-cleaving activity of resveratrol in the presence of Cu(II)

Kiyoshi Fukuhara, Maki Nagakawa, Ikuo Nakanishi, Kei Ohkubo, Kohei Imai, Shiro Urano, Shunichi Fukuzumi, Toshihiko Ozawa, Nobuo Ikota, Masataka Mochizuki, Naoki Miyata, Haruhiro Okuda

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 210 KB

english, 2006

16

Polyamine conjugates of meso-tritolylporphyrin and protoporphyrin IX: Potential agents for photodynamic therapy of cancers

Vincent Sol, François Lamarche, Michaela Enache, Guillaume Garcia, Robert Granet, Michel Guilloton, J.C. Blais, Pierre Krausz

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 440 KB

english, 2006

17

Classification of dopamine antagonists using functional feature hypothesis and topological descriptors

Hye-Jung Kim, Yong Seo Cho, Hun Yeong Koh, Jae Yang Kong, Kyoung Tai No, Ae Nim Pae

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 543 KB

english, 2006

18

Understanding the structure–activity and structure–selectivity correlation of cyclic guanine derivatives as phosphodiesterase-5 inhibitors by molecular docking, CoMFA and CoMSIA analyses

Guang-Fu Yang, Hai-Ting Lu, Ying Xiong, Chang-Guo Zhan

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 815 KB

english, 2006

19

A combined approach of docking and 3D QSAR study of β-ketoacyl-acyl carrier protein synthase III (FabH) inhibitors

Ali Ashek, Seung Joo Cho

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 634 KB

english, 2006

20

Substituted phenanthrenes with basic amino side chains: A new series of anti-breast cancer agents

Shagufta, Ajay Kumar Srivastava, Ramesh Sharma, Rajeev Mishra, Anil Kumar Balapure, Puvvada S.R. Murthy, Gautam Panda

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 325 KB

english, 2006

21

3D-QSAR studies on tripeptide aldehyde inhibitors of proteasome using CoMFA and CoMSIA methods

Yong-Qiang Zhu, Jian-Feng Pei, Zhen-Ming Liu, Lu-Hua Lai, Jing-Rong Cui, Run-Tao Li

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 866 KB

english, 2006

22

Modelling, synthesis and biological evaluation of novel glucuronide-based probes of Vibrio cholerae sialidase

Maretta C. Mann, Robin J. Thomson, Jeffrey C. Dyason, Sarah McAtamney, Mark von Itzstein

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 486 KB

english, 2006

23

Synthesis of chalcone analogues with increased antileishmanial activity

Paula Boeck, Camila Alves Bandeira Falcão, Paulo César Leal, Rosendo Augusto Yunes, Valdir Cechinel Filho, Eduardo Caio Torres-Santos, Bartira Rossi-Bergmann

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 205 KB

english, 2006

24

DFT study of the reductive decomposition of artemisinin

Alex Gutterres Taranto, José Walkimar de Mesquita Carneiro, Martha Teixeira de Araujo

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 678 KB

english, 2006

25

Theoretical proton affinities of α1 adrenoceptor ligands

Gemma K. Kinsella, Graeme W. Watson, Isabel Rozas

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 148 KB

english, 2006

26

Direct observation (NMR) of the efficacy of glucagon receptor antagonists in murine liver expressing the human glucagon receptor

Sheila M. Cohen, Joseph L. Duffy, Corin Miller, Brian A. Kirk, Mari Rios Candelore, Victor D.H. Ding, Gregory Kaczorowski, Laurie M. Tota, Jeffrey G. Werrmann, Michael Wright, Emma R. Parmee, James R.

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 462 KB

english, 2006

27

Synthesis and biological evaluation of a series of flavone derivatives as potential radioligands for imaging the multidrug resistance-associated protein 1 (ABCC1/MRP1)

Sylvie Mavel, Branko Dikic, Somchit Palakas, Patrick Emond, Ivan Greguric, Adrienne Gomez de Gracia, Filomena Mattner, Manuel Garrigos, Denis Guilloteau, Andrew Katsifis

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 177 KB

english, 2006

28

The development of 3D-QSAR study and recursive partitioning of heterocyclic quinone derivatives with antifungal activity

Su-Young Choi, Jae Hong Shin, Chung Kyu Ryu, Ky-Youb Nam, Kyoung Tai No, Hea-Young Park Choo

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 360 KB

english, 2006

29

Solid phase synthesis and antiprotozoal evaluation of di- and trisubstituted 5′-carboxamidoadenosine analogues

Boris Rodenko, Remko J. Detz, Victorine A. Pinas, Catia Lambertucci, Reto Brun, Martin J. Wanner, Gerrit-Jan Koomen

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 292 KB

english, 2006

30

Advances in the synthesis and recent therapeutic applications of 1,2,4-thiadiazole heterocycles

Ana Castro, Tania Castaño, Arantxa Encinas, Williams Porcal, Carmen Gil

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 213 KB

english, 2006

31

Evaluation of aldose reductase inhibition and docking studies of some secondary metabolites, isolated from Origanum vulgare L. ssp. hirtum

Catherine Koukoulitsa, Chariklia Zika, George D. Geromichalos, Vassilis J. Demopoulos, Helen Skaltsa

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 518 KB

english, 2006

32

3D QSAR study of hypolipidemic asarones by comparative molecular surface analysis

Tomasz Magdziarz, Bozena Łozowicka, Rafał Gieleciak, Andrzej Bąk, Jarosław Polański, Zdzisław Chilmonczyk

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 930 KB

english, 2006

33

In vitro oxidative metabolism study of (−)-rhazinilam

Anne Décor, Delphine Bellocq, Odile Thoison, Nicolas Lekieffre, Angèle Chiaroni, Jamal Ouazzani, Thierry Cresteil, Françoise Guéritte, Olivier Baudoin

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 261 KB

english, 2006

34

Studies of interaction of trichloro{η2-cis-N,N-dimethyl-1-[6-(N′,N′-dimethyl-ammoniummethyl)-cyclohex-3-ene-1-yl]-methylammonium}platinum(II) chloride with DNA: Effects on secondary and tertiary structures of DNA. Cytotoxic assays on human ovarian cancer cell lines, resistant and non-resistant to cisplatin

Marina Gay, Ángel M. Montaña, Virtudes Moreno, María-José Prieto, José Manuel Pérez, Carlos Alonso

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 316 KB

english, 2006

35

Synthesis and biological evaluation of 9-(5′,5′-difluoro-5′-phosphonopentyl)guanine derivatives for PNP-inhibitors

Sadao Hikishima, Machiko Isobe, Satoru Koyanagi, Shinji Soeda, Hiroshi Shimeno, Shiroshi Shibuya, Tsutomu Yokomatsu

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 235 KB

english, 2006

36

Structure–activity relationships of a series of tariquidar analogs as multidrug resistance modulators

Christoph Globisch, Ilza K. Pajeva, Michael Wiese

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 581 KB

english, 2006

37

Activity of lupane triterpenoids from Maytenus species as inhibitors of nitric oxide and prostaglandin E2

Carolina P. Reyes, Marvin J. Núñez, Ignacio A. Jiménez, Jérôme Busserolles, María J. Alcaraz, Isabel L. Bazzocchi

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 165 KB

english, 2006

38

Corrigendum to “Molecular modeling and 3D-QSAR studies of indolomorphinan derivatives as kappa opioid antagonists” [Bioorg. Med. Chem. 14 (2006) 601–610]

Wei Li, Yun Tang, You-Li Zheng, Zhui-Bai Qiu

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Fichier:

PDF, 57 KB

2006

39

Instructions to contributors

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 32 KB

english, 2006

40

Editorial Board

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 315 KB

english, 2006

41

Graphical contents list

Journal:

Bioorganic & Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 306 KB

english, 2006