Volume 13; Issue 16

Bioorganic & Medicinal Chemistry

Volume 13; Issue 16

1

Preventive effects of soyasapogenol B derivatives on liver injury in a concanavalin A-induced hepatitis model

Kazue Sasaki, Nobuto Minowa, Hiroyuki Kuzuhara, Shoji Nishiyama

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 334 KB

english, 2005

2

Design and synthesis of low molecular weight compounds with complement inhibition activity

Hoshang E. Master, Shabana I. Khan, Krishna A. Poojari

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 516 KB

english, 2005

3

Genistein derivatives as selective estrogen receptor modulators: Sonochemical synthesis and in vivo anti-osteoporotic action

Shi F. Wang, Qing Jiang, Yong H. Ye, Yang Li, Ren X. Tan

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 810 KB

english, 2005

4

Design, synthesis, and biological evaluation of novel naphthoquinone derivatives with CDC25 phosphatase inhibitory activity

Marie-Priscille Brun, Emmanuelle Braud, Delphine Angotti, Odile Mondésert, Muriel Quaranta, Matthieu Montes, Maria Miteva, Nohad Gresh, Bernard Ducommun, Christiane Garbay

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 476 KB

english, 2005

5

Novel thiazonaphthalimides as efficient antitumor and DNA photocleaving agents: Effects of intercalation, side chains, and substituent groups

Zhigang Li, Qing Yang, Xuhong Qian

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 788 KB

english, 2005

6

A new structural alternative in benzo[b]furans for antimicrobial activity

M. Wahab Khan, M. Jahangir Alam, M.A. Rashid, R. Chowdhury

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 369 KB

english, 2005

7

Protonated structures of naturally occurring deoxyribonucleic acids and their interaction with berberine

Kakali Bhadra, Gopinatha Suresh Kumar, Suman Das, Md. Maidul Islam, Motilal Maiti

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 572 KB

english, 2005

8

Synthesis of novel 5-aryl-2-thio-1,3,4-oxadiazoles and the study of their structure–anti-mycobacterial activities

Fliur Macaev, Ghenadie Rusu, Serghei Pogrebnoi, Alexandru Gudima, Eugenia Stingaci, Ludmila Vlad, Nathaly Shvets, Fatma Kandemirli, Anatholy Dimoglo, Robert Reynolds

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 417 KB

english, 2005

9

RO4383596, an orally active KDR, FGFR, and PDGFR inhibitor: Synthesis and biological evaluation

Lee A. McDermott, Mary Simcox, Brian Higgins, Tom Nevins, Kenneth Kolinsky, Melissa Smith, Hong Yang, Jia K. Li, Yingsi Chen, June Ke, Navita Mallalieu, Tom Egan, Stan Kolis, Aruna Railkar, Louise Ger

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 367 KB

english, 2005

10

Insight into 2-phenylpyrazolo[1,5-a]pyrimidin-3-yl acetamides as peripheral benzodiazepine receptor ligands: Synthesis, biological evaluation and 3D-QSAR investigation

Silvia Selleri, Paola Gratteri, Camilla Costagli, Claudia Bonaccini, Annarella Costanzo, Fabrizio Melani, Gabriella Guerrini, Giovanna Ciciani, Barbara Costa, Francesca Spinetti, Claudia Martini, Fabr

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 1.20 MB

english, 2005

11

Oligonucleotides containing 2′-O-[2-(2,3-dihydroxypropyl)amino-2-oxoethyl]uridine as suitable precursors of 2′-aldehyde oligonucleotides for chemoselective ligation

Eugeny M. Zubin, Dmitry A. Stetsenko, Timofei S. Zatsepin, Michael J. Gait, Tatiana S. Oretskaya

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 355 KB

english, 2005

12

Efficient synthesis of fluorothiosparfosic acid analogues with potential antitumoral activity

Emmanuel Pfund, Thierry Lequeux, Serge Masson, Michel Vazeux, Alex Cordi, Alain Pierre, Valérie Serre, Guy Hervé

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 277 KB

english, 2005

13

Lewis acid-promoted transformation of 2-alkoxypyridines into 2-aminopyridines and their antibacterial activity. Part 2: Remarkably facile C–N bond formation

Alaa A.-M. Abdel-Aziz, Hussein I. El-Subbagh, Takehisa Kunieda

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 472 KB

english, 2005

14

Syntheses and binding affinities of 6-nitroquipazine analogues for serotonin transporter. Part 4: 3-Alkyl-4-halo-6-nitroquipazines

Byung Seok Moon, Byoung Se Lee, Dae Yoon Chi

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 251 KB

english, 2005

15

Synthetic studies on novel Syk inhibitors. Part 1: Synthesis and structure–activity relationships of pyrimidine-5-carboxamide derivatives

Hiroyuki Hisamichi, Ryo Naito, Akira Toyoshima, Noriyuki Kawano, Atsushi Ichikawa, Akiko Orita, Masaya Orita, Noritaka Hamada, Makoto Takeuchi, Mitsuaki Ohta, Shin-ichi Tsukamoto

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 842 KB

english, 2005

16

Geldanamycin derivative inhibition of HGF/SF-mediated Met tyrosine kinase receptor-dependent urokinase-plasminogen activation

Yuehai Shen, Qian Xie, Monica Norberg, Edward Sausville, George Vande Woude, David Wenkert

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 291 KB

english, 2005

17

Novel 3-amino-2-hydroxy acids containing protease inhibitors. Part 1: Synthesis and kinetic characterization as aminopeptidase P inhibitors

Angela Stöckel-Maschek, Beate Stiebitz, Regine Koelsch, Klaus Neubert

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 512 KB

english, 2005

18

Editorial Board

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 209 KB

english, 2005

19

Graphical contents list

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 597 KB

english, 2005

20

Contributors to this issue

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Fichier:

PDF, 183 KB

2005

21

Instructions to contributors

Journal:

Bioorganic & Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 32 KB

english, 2005