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Volume 84; Issue 1
Main
Biochemical Pharmacology
Volume 84; Issue 1
Biochemical Pharmacology
Volume 84; Issue 1
1
Searching for molecular targets in sarcoma
Beverly A. Teicher
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 433 KB
Vos balises:
english, 2012
2
Complex roles of members of the ADP-ribosyl transferase super family in immune defences: Looking beyond PARP1
Iain Welsby
,
David Hutin
,
Oberdan Leo
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 678 KB
Vos balises:
english, 2012
3
Allopurinol, quercetin and rutin ameliorate renal NLRP3 inflammasome activation and lipid accumulation in fructose-fed rats
Qing-Hua Hu
,
Xian Zhang
,
Ying Pan
,
Yu-Cheng Li
,
Ling-Dong Kong
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 1.75 MB
Vos balises:
english, 2012
4
Discovery of novel A3 adenosine receptor ligands based on chromone scaffold
Alexandra Gaspar
,
Joana Reis
,
Sonja Kachler
,
Silvia Paoletta
,
Eugenio Uriarte
,
Karl-Norbert Klotz
,
Stefano Moro
,
Fernanda Borges
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 678 KB
Vos balises:
english, 2012
5
The role of the second and third extracellular loops of the adenosine A1 receptor in activation and allosteric modulation
M.C. Peeters
,
L.E. Wisse
,
A. Dinaj
,
B. Vroling
,
G. Vriend
,
A.P. IJzerman
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 1.26 MB
Vos balises:
english, 2012
6
Inhibition of thymidine phosphorylase expression by using an HSP90 inhibitor potentiates the cytotoxic effect of cisplatin in non-small-cell lung cancer cells
Shao-Hsing Weng
,
Sheng-Chieh Tseng
,
Yu-Ching Huang
,
Huang-Jen Chen
,
Yun-Wei Lin
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 2.32 MB
Vos balises:
english, 2012
7
Binding and activity of the prostacyclin receptor (IP) agonists, treprostinil and iloprost, at human prostanoid receptors: Treprostinil is a potent DP1 and EP2 agonist
Brendan J. Whittle
,
Adam M. Silverstein
,
David M. Mottola
,
Lucie H. Clapp
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 392 KB
Vos balises:
english, 2012
8
Diminished toxicity of C-1748, 4-methyl-9-hydroxyethylamino-1-nitroacridine, compared with its demethyl analog, C-857, corresponds to its resistance to metabolism in HepG2 cells
Anita Wiśniewska
,
Magdalena Niemira
,
Karolina Jagiełło
,
Agnieszka Potęga
,
Małgorzata Świst
,
Colin Henderson
,
Anna Skwarska
,
Ewa Augustin
,
Jerzy Konopa
,
Zofia Mazerska
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 1.29 MB
Vos balises:
english, 2012
9
Estradiol induces cytochrome P450 2B6 expression at high concentrations: Implication in estrogen-mediated gene regulation in pregnancy
Kwi Hye Koh
,
Steve Jurkovic
,
Kyunghee Yang
,
Su-Young Choi
,
Jin Woo Jung
,
Kwang Pyo Kim
,
Wei Zhang
,
Hyunyoung Jeong
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 1.29 MB
Vos balises:
english, 2012
10
Intestinal CYP3A4 and midazolam disposition in vivo associate with VDR polymorphisms and show seasonal variation
Ranjit K. Thirumaran
,
Jatinder K. Lamba
,
Richard B. Kim
,
Brad L. Urquhart
,
Jamie C. Gregor
,
Nilesh Chande
,
Yiping Fan
,
An Qi
,
Cheng Cheng
,
Kenneth E. Thummel
,
Stephen D. Hall
,
Erin G. Schuetz
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 478 KB
Vos balises:
english, 2012
11
Eriodictyol prevents early retinal and plasma abnormalities in streptozotocin-induced diabetic rats
Claudio Bucolo
,
Gian Marco Leggio
,
Filippo Drago
,
Salvatore Salomone
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 395 KB
Vos balises:
english, 2012
12
The anticancer thiosemicarbazones Dp44mT and triapine lack inhibitory effects as catalytic inhibitors or poisons of DNA topoisomerase IIα
Jack C. Yalowich
,
Xing Wu
,
Rui Zhang
,
Ragu Kanagasabai
,
Marisa Hornbaker
,
Brian B. Hasinoff
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 585 KB
Vos balises:
english, 2012
13
Phosphorylation of deoxycytidine kinase on Ser-74: Impact on kinetic properties and nucleoside analog activation in cancer cells
Rachid Amsailale
,
Eric Van Den Neste
,
Angélique Arts
,
Eliza Starczewska
,
Françoise Bontemps
,
Caroline Smal
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 693 KB
Vos balises:
english, 2012
14
Rottlerin potentiates camptothecin-induced cytotoxicity in human hormone refractory prostate cancers through increased formation and stabilization of topoisomerase I-DNA cleavage complexes in a PKCδ-independent pathway
Jui-Ling Hsu
,
Yunn-Fang Ho
,
Tsai-Kun Li
,
Ching-Shih Chen
,
Lih-Ching Hsu
,
Jih-Hwa Guh
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 1.43 MB
Vos balises:
english, 2012
15
Editorial Advisory Board
Journal:
Biochemical Pharmacology
Année:
2012
Langue:
english
Fichier:
PDF, 35 KB
Vos balises:
english, 2012
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