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Volume 80; Issue 9
Main
Biochemical Pharmacology
Volume 80; Issue 9
Biochemical Pharmacology
Volume 80; Issue 9
1
Activation of the p38 pathway by a novel monoketone curcumin analog, EF24, suggests a potential combination strategy
Shala L. Thomas
,
Jing Zhao
,
Zijian Li
,
Bin Lou
,
Yuhong Du
,
Jamie Purcell
,
James P. Snyder
,
Fadlo R. Khuri
,
Dennis Liotta
,
Haian Fu
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 371 KB
Vos balises:
english, 2010
2
Glycine transporter (GlyT1) inhibitors with reduced residence time increase prepulse inhibition without inducing hyperlocomotion in DBA/2 mice
Karla Kopec
,
Dorothy G. Flood
,
Maciej Gasior
,
Beth Ann W. McKenna
,
Eva Zuvich
,
Justin Schreiber
,
Joseph M. Salvino
,
John T. Durkin
,
Mark A. Ator
,
Michael J. Marino
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 501 KB
Vos balises:
english, 2010
3
Conformational flexibility of transmembrane helix VII of the human serotonin transporter impacts ion dependence and transport
Cody J. Wenthur
,
Gustavo J. Rodríguez
,
Charles P. Kuntz
,
Eric L. Barker
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 468 KB
Vos balises:
english, 2010
4
The rGel/BLyS fusion toxin inhibits STAT3 signaling via down-regulation of interleukin-6 receptor in diffuse large B-cell lymphoma
Mi-Ae Lyu
,
Bokyung Sung
,
Lawrence H. Cheung
,
John W. Marks
,
Bharat B. Aggarwal
,
Ricardo C.T. Aguiar
,
Michael G. Rosenblum
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 386 KB
Vos balises:
english, 2010
5
Serine phosphorylation of glutathione S-transferase P1 (GSTP1) by PKCα enhances GSTP1-dependent cisplatin metabolism and resistance in human glioma cells
Simendra Singh
,
Tatsunori Okamura
,
Francis Ali-Osman
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 619 KB
Vos balises:
english, 2010
6
Y124 at the peripheral anionic site is important for the reactivation of nerve agent-inhibited acetylcholinesterase by H oximes
Chunyuan Luo
,
Carolyn Chambers
,
Nagarajan Pattabiraman
,
Min Tong
,
Prasanthi Tipparaju
,
Ashima Saxena
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 812 KB
Vos balises:
english, 2010
7
Quantitative relationship between guanine O6-alkyl lesions produced by Onrigin™ and tumor resistance by O6-alkylguanine-DNA alkyltransferase
Kimiko Ishiguro
,
Yong-Lian Zhu
,
Krishnamurthy Shyam
,
Philip G. Penketh
,
Raymond P. Baumann
,
Alan C. Sartorelli
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 356 KB
Vos balises:
english, 2010
8
Modulation of HDL metabolism by the niacin receptor GPR109A in mouse hepatocytes
Xiaoyu Li
,
John S. Millar
,
Nicholas Brownell
,
François Briand
,
Daniel J. Rader
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 559 KB
Vos balises:
english, 2010
9
Glutamine as a mediator of ammonia neurotoxicity: A critical appraisal
Jan Albrecht
,
Magdalena Zielińska
,
Michael D. Norenberg
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 218 KB
Vos balises:
english, 2010
10
Polo-like kinase1 (Plk1) knockdown enhances cisplatin chemosensitivity via up-regulation of p73α in p53 mutant human epidermoid squamous carcinoma cells
Shilpa Tyagi
,
Kulpreet Bhui
,
Richa Singh
,
Madhulika Singh
,
Sheikh Raisuddin
,
Yogeshwer Shukla
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 575 KB
Vos balises:
english, 2010
11
Inhibition of cell growth and potentiation of tumor necrosis factor-α (TNF-α)-induced apoptosis by a phenanthroindolizidine alkaloid antofine in human colon cancer cells
Hye-Young Min
,
Hwa-Jin Chung
,
Eun-Hye Kim
,
Sanghee Kim
,
Eun-Jung Park
,
Sang Kook Lee
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 475 KB
Vos balises:
english, 2010
12
Comparison of the pharmacological properties of human and rat histamine H3-receptors
David Schnell
,
Andrea Strasser
,
Roland Seifert
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 889 KB
Vos balises:
english, 2010
13
Newly synthetic ceramide-1-phosphate analogs; their uptake, intracellular localization, and roles as an inhibitor of cytosolic phospholipase A2α and inducer of cell toxicity
Tomohiko Makiyama
,
Nobuo Nagasaka
,
Yuuya Houjyo
,
Erika Yamaura
,
Hiroyuki Nakamura
,
Yuuki Koide
,
Atsushi Nishida
,
Toshihiko Murayama
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 1.80 MB
Vos balises:
english, 2010
14
Dimethylcelecoxib inhibits mPGES-1 promoter activity by influencing EGR1 and NF-κB
Klaus Deckmann
,
Florian Rörsch
,
Ramona Steri
,
Manfred Schubert-Zsilavecz
,
Gerd Geisslinger
,
Sabine Grösch
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 395 KB
Vos balises:
english, 2010
15
Chain-dependent photocytotoxicity of tricationic porphyrin conjugates and related mechanisms of cell death in proliferating human skin keratinocytes
João Nuno Silva
,
Antoine Galmiche
,
João P.C. Tomé
,
Agnès Boullier
,
Maria G.P.M.S. Neves
,
Eduarda M.P. Silva
,
Jean-Claude Capiod
,
José A.S. Cavaleiro
,
René Santus
,
Jean-Claude Mazière
,
Paulo Filipe
,
Pa
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 1.43 MB
Vos balises:
english, 2010
16
Resveratrol modulates angiogenesis through the GSK3β/β-catenin/TCF-dependent pathway in human endothelial cells
Hui Wang
,
Haibin Zhou
,
Yongxin Zou
,
Qiao Liu
,
Chenhong Guo
,
Guimin Gao
,
Changshun Shao
,
Yaoqin Gong
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 1.02 MB
Vos balises:
english, 2010
17
Editorial Advisory Board
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 31 KB
Vos balises:
english, 2010
18
Graphical Abstracts Contents
Journal:
Biochemical Pharmacology
Année:
2010
Langue:
english
Fichier:
PDF, 828 KB
Vos balises:
english, 2010
1
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