Volume 38; Issue 5

Journal of Medicinal Chemistry

Volume 38; Issue 5

1

Synthesis and Anti-HIV-1 Activity of 4,5,6,7-Tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one (TlBO) Derivatives. 4

Ho, Winston, Kukla, Michael J., Breslin, Henry J., Ludovici, Donald W., Grous, Philip P., Diamond, Craig J., Miranda, Milton, Rodgers, James D., Ho, Chih Y.

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 1.19 MB

english, 1995

2

Fluorine for Hydroxy Substitution in Biogenic Amines: Asymmetric Synthesis and Biological Evaluation of Fluorine-18-Labeled .beta.-Fluorophenylalkylamines as Model Systems

Dort, Marcian E. Van, Jung, Yong-Woon, Sherman, Philip S., Kilbourn, Michael R., Wieland, Donald M.

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 828 KB

english, 1995

3

[[[(Thienylcarbonyl)alkyl]oxy]phenyl]- and [[[(Pyrrylcarbonyl)alkyl]oxy]phenyl]oxazoline Derivatives with Potent and Selective Antihuman Rhinovirus Activity

Massa, Silvio, Corelli, Federico, Artico, Marino, Mai, Antonello, Ragno, Rino, De Montis, Antonella, Loi, Anna Giulia, Corrias, Simona, Marongiu, Maria Elena, La Colla, Paolo

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 767 KB

english, 1995

4

Chemically Stable N-Methyl-4-(alkylthio)cyclophosphamide Derivatives as Prodrugs of 4-Hydroxycyclophosphamide

Moon, Ki-Young, Shirota, Frances N., Baturay, Nesrine, Kwon, Chul-Hoon

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 590 KB

english, 1995

5

Synthesis and Anti-HIV-1 Activity of 4,5,6,7-Tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one (TIBO) Derivatives. 3

Breslin, Henry J., Kukla, Michael J., Ludovici, Donald W., Mohrbacher, Richard, Ho, Winston, Miranda, Milton, Rodgers, James D., Hitchens, T. Kevin, Leo, Gregory

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 3.03 MB

english, 1995

6

Synthesis of 11.beta.-[18F]Fluoro-5.alpha.-dihydrotestosterone and 11.beta.-[18F]Fluoro-19-nor-5.alpha.-dihydrotestosterone: Preparation via Halofluorination-Reduction, Receptor Binding, and Tissue Distribution

Choe, Yearn Seong, Lidstroem, Pelle J., Chi, Dae Yoon, Bonasera, Thomas A., Welch, Michael J., Katzenellenbogen, John A.

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 1.37 MB

english, 1995

7

2,4-Diamino-5-substituted-quinazolines as Inhibitors of a Human Dihydrofolate Reductase with a Site-Directed Mutation at Position 22 and of the Dihydrofolate Reductases from Pneumocystis carinii and Toxoplasma gondii

Rosowsky, Andre, Mota, Clara E., Queener, Sherry F., Waltham, Mark, Ercikan-Abali, Emine, Bertino, Joseph R.

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 1.13 MB

english, 1995

8

Structural and Conformational Requirements for Human Calcitonin Activity: Design, Synthesis, and Study of Lactam-Bridged Analogs

Kapurniotu, Afrodite, Taylor, John W.

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 2.31 MB

english, 1995

9

Orally Bioavailable Benzisothiazolone Inhibitors of Human Leukocyte Elastase

Hlasta, Dennis J., Subramanyam, Chakrapani, Bell, Malcolm R., Carabateas, Philip M., Court, John J., Desai, Ranjit C., Drozd, Marion L., Eickhoff, W. Mark, Ferguson, Edward W., Gordon, Robert J., Dunl

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 752 KB

english, 1995

10

Antimalarial Activity of New Dihydroartemisinin Derivatives. 6. .alpha.-Alkylbenzylic Ethers

Lin, Ai Jeng, Miller, Robert E.

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 726 KB

english, 1995

11

Synthesis, Biological Evaluation, and Structure Analysis of a Series of New 1,5-Anhydrohexitol Nucleosides

Verheggen, Ilse, Van Aerschot, Arthur, Van Meervelt, Luc, Rozenski, Jef, Wiebe, Leonard, Snoeck, Robert, Andrei, Graciela, Balzarini, Jan, Claes, Paul

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 1.48 MB

english, 1995

12

Book Reviews

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 298 KB

english, 1995

13

Masthead

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 175 KB

english, 1995

14

Structure-Activity Studies of 2,3,4,4a,5,9b-Hexahydroindeno[1,2-c]pyridines as Antispermatogenic Agents for Male Contraception

Cook, C. Edgar, Wani, Mansukh C., Jump, Joseph M., Lee, Yue-W., Fail, Patricia A., Anderson, Stephanie A., Gu, Yu-Q., Petrow, Vladimir

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 1.29 MB

english, 1995