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Volume 37; Issue 7

Journal of Medicinal Chemistry

Volume 37; Issue 7

1

A Novel 3-Substituted Benzazepinone Growth Hormone Secretagogue (L-692,429)

Prendergast, Kristine, Wyvratt, Matthew J., Fisher, Michael H., Cheng, Kang, Chan, Wanda W.-S., Butler, Bridget, Smith, Roy G., Ball, Richard G., Schoen, William R., Pisano, Judith M.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 2.02 MB

english, 1994

2

Homodimeric and Heterodimeric Bis(amino thiol) Oxometal Complexes with Rhenium(V) and Technetium(V). Control of Heterodimeric Complex Formation and an Approach to Metal Complexes that Mimic Steroid Hormones

Chi, Dae Yoon, O'Neil, James P., Anderson, Carolyn J., Welch, Michael J., Katzenellenbogen, John A.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.52 MB

english, 1994

3

Discovery, Synthesis, and Bioactivity of Bis(heteroaryl)piperazines. 1. A Novel Class of Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors

Romero, Donna L., Morge, Raymond A., Biles, Carolyn, Berrios-Pena, Norman, May, Paul D., Palmer, John R., Johnson, Paul D., Smith, Herman W., Busso, Mariano, et. al.,

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 2.34 MB

english, 1994

4

Benzoxazolamines and Benzothiazolamines: Potent, Enantioselective Inhibitors of Leukotriene Biosynthesis with a Novel Mechanism of Action

Lazer, Edward S., Miao, Clara K., Wong, Hin-Chor, Sorcek, Ronald, Spero, Denice M., Gilman, Alex, Pal, Kollol, Behnke, Mark, Graham, Anne G.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.46 MB

english, 1994

5

Guaiacoxypropanolamine Derivatives of Capsaicin: A New Family of .beta.-Adrenoceptor Blockers with Intrinsic Cardiotonic Properties

Chen, Ing-Jun, Yeh, Jwu-Lai, Liou, Shwu-Jen, Shen, Ai-Yu

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 813 KB

english, 1994

6

Antiinflammatory 4,5-Diarylpyrroles: Synthesis and QSAR

Wilkerson, Wendell W., Galbraith, William, Gans-Brangs, Kathleen, Grubb, Mary, Hewes, Walter E., Jaffee, Bruce, Kenney, J. P., Kerr, Janet, Wong, Nancy

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.48 MB

english, 1994

7

Synthesis of L-Thiocitrulline, L-Homothiocitrulline, and S-Methyl-L-thiocitrulline: A New Class of Potent Nitric Oxide Synthase Inhibitors

Narayanan, Krishnaswamy, Griffith, Owen W.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 443 KB

english, 1994

8

Enkephalin Analogs as Systemically Active Antinociceptive Agents: O- and N-Alkylated Derivatives of the Dipeptide Amide L-2,6-Dimethyltyrosyl-N-(3-phenylpropyl)-D-alaninamide

Pitzele, Barnett S., Hamilton, Robert W., Kudla, Kathleen D., Tsymbalov, Sofya, Stapelfeld, Awilda, Savage, Michael A., Clare, Michael, Hammond, Donna L., Hansen, Donald W.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.16 MB

english, 1994

9

Iron(III)-Chelating Resins. IX. Antibacterial Activity of a Water-Insoluble Iron(III)-Chelating Resin

Feng, Minhua, van der Does, Leen, Bantjes, Adriaan

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 903 KB

english, 1994

10

6H-Pyrazolo[4,5,1-de]acridin-6-ones as a Novel Class of Antitumor Agents.Synthesis and Biological Activity

Sugaya, Toru, Mimura, Yukiteru, Shida, Yasusi, Osawa, Yutaka, Matsukuma, Ikuo, Ikeda, Shunichi, Akinaga, Shiro, Morimoto, Makoto, Ashizawa, Tadashi

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 624 KB

english, 1994

11

Structure-based design of inhibitors of purine nucleoside phosphorylase. 3. 9-Arylmethyl derivatives of 9-deazaguanine substituted on the arylmethyl group. [Erratum to document cited in CA119(25):271601v]

Erion, Mark D., Niwas, Shri, Rose, Jerry D., Ananthan, Subramaniam, Allen, Mark, Secrist, John A., Babu, Y. Sudhakar, Bugg, Charles E., Guida, Wayne C.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 50 KB

english, 1994

12

A Nonlinear Map of Substituent Constants for Selecting Test Series and Deriving Structure-Activity Relationships. I. Aromatic Series

Domine, Daniel, Devillers, James, Chastrette, Maurice

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 999 KB

english, 1994

13

A Nonlinear Map of Substituent Constants for Selecting Test Series and Deriving Structure-Activity Relationships. II. Aliphatic Series

Domine, Daniel, Devillers, James, Chastrette, Maurice

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 792 KB

english, 1994

14

Specific Inhibitors of Ileal Bile Acid Transport

Wess, Guenther, Kramer, Werner, Enhsen, Alfons, Glombik, Heiner, Baringhaus, Karl-Heinz, Boeger, Georg, Urmann, Matthias, Bock, Klaus, Kleine, Horst

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 262 KB

english, 1994

15

Dianilinophthalimides: Potent and Selective, ATP-Competitive Inhibitors of the EGF-Receptor Protein Tyrosine Kinase

Trinks, Uwe, Buchdunger, Elisabeth, Furet, Pascal, Kump, Wilhelm, Mett, Helmut, Meyer, Thomas, Mueller, Marcel, Regenass, Urs, Rihs, Greti

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 2.49 MB

english, 1994

16

Resolution, Absolute Stereochemistry, and Pharmacology of the S-(+)- and R-(-)-Isomers of the Apparent Partial AMPA Receptor Agonist (R,S)-2-Amino-3-(3-hydroxy-5-phenylisoxazol-4-yl)propionic Acid [(R,S)-APPA]

Ebert, Bjarke, Lenz, Sibylle, Brehm, Lotte, Bregnedal, Peter, Hansen, Jan J., Frederiksen, Kristen, Bogeso, Klaus P., Krogsgaard-Larsen, Povl

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 858 KB

english, 1994

17

Synthesis of Selective Non-Ca2+ Mobilizing Inhibitors of D-myo-Inositol 1,4,5-Trisphosphate 5-Phosphatase

Lampe, Dethard, Liu, Changsheng, Potter, Barry V. L.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 928 KB

english, 1994

18

The Use of the GRID Program in the 3-D QSAR Analysis of a Series of Calcium-Channel Agonists

Davis, Andrew M., Gensmantel, Nigel P., Johansson, Erik, Marriott, David P.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 3.59 MB

english, 1994

19

Book Reviews

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 92 KB

english, 1994

20

A new orally active insulin-mimetic vanadyl complex: bis(pyrrolidine-N-carbodithioato)oxovanadium(IV)

Watanabe, Hiromi, Nakai, Masami, Komazawa, Kyoko, Sakurai, Hiromu

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 803 KB

english, 1994

21

Development of a Receptor-Interaction Model for Serotonin 5-HT2 Receptor Antagonists. Predicting Selectivity with Respect to Dopamine D2 Receptors

Andersen, Kim, Liljefors, Tommy, Gundertofte, Klaus, Perregaard, Jens, Bogeso, Klaus P.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 3.19 MB

english, 1994

22

Novel 4-(Aryloxy)tetrahydropyridine Analogs of MPTP as Monoamine Oxidase A and B Substrates

Kalgutkar, Amit S., Castagnoli, Kay, Hall, Andrea, Castagnoli, Neal

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 810 KB

english, 1994

23

Masthead

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 174 KB

english, 1994

24

Non-peptide angiotensin II receptor antagonists. 2. Design, synthesis, and biological activity of N-substituted (phenylamino)phenylacetic acids and acyl sulfonamides. [Erratum to document cited in CA120(5):45190z]

Dhanoa, Daljit S., Bagley, Scott W., Chang, Raymond S. L., Lotti, Victor J., Chen, Tsing Bau, Kivlighn, Salah D., Zingaro, Gloria J., Siegl, Peter K. S., Patchett, Arthur A., Greenlee, William J.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 50 KB

english, 1994