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Volume 37; Issue 16

Journal of Medicinal Chemistry

Volume 37; Issue 16

1

Non-Peptide Fibrinogen Receptor Antagonists. 2. Optimization of a Tyrosine Template as a Mimic for Arg-Gly-Asp

Egbertson, Melissa S., Chang, Charles T.-C., Duggan, Mark E., Gould, Robert J., Halczenko, Wasyl, Hartman, George D., Laswell, William L., Lynch, Joseph J., Lynch, Robert J.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 2.44 MB

english, 1994

2

Cyclic Benzamides as Mixed Dopamine D2/Serotonin 5-HT2 Receptor Antagonists: Potential Atypical Antipsychotic Agents

Norman, Mark H., Rigdon, Greg C., Navas, Frank, Cooper, Barrett R.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.83 MB

english, 1994

3

Synthesis and Pharmacological Properties of 11-Hydroxy-3-(1',1'-dimethylheptyl)hexahydrocannabinol: A High Affinity Cannabinoid Agonist

Yan, Guo, Yin, Dali, Khanolkar, Atmaram D., Compton, David R., Martin, Billy R., Makriyannis, Alexandros

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 405 KB

english, 1994

4

5-[(3-Nitropyrid-2-yl)amino]indoles: Novel Serotonin Agonists with Selectivity for the 5-HT1D Receptor. Variation of the C3 Substituent on the Indole Template Leads to Increased 5-HT1D Receptor Selectivity

Macor, John E., Blank, David H., Fox, Carol B., Lebel, Lorraine A., Newman, Michael E., Post, Ronald J., Ryan, Kevin, Schmidt, Anne W., Schulz, David W., Koe, B. Kenneth

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 498 KB

english, 1994

5

Masthead

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 170 KB

english, 1994

6

HIV-1 Reverse Transcriptase Inhibitor Design Using Artificial Neural Networks

Tetko, Igor V., Tanchuk, Vsevolod Yu., Chentsova, Neliya P., Antonenko, Svetlana V., Poda, Gennady I., Kukhar, Valery P., Luik, Alexander I.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 732 KB

english, 1994

7

Spirovesamicols: Conformationally Restricted Analogs of 2-(4-Phenylpiperidino)cyclohexanol (Vesamicol, AH5183) as Potential Modulators of Presynaptic Cholinergic Function

Efange, S. M. N., Khare, A. B., Foulon, C., Akella, S. K., Parsons, S. M.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.29 MB

english, 1994

8

Comparative Molecular Field Analysis Using GRID Force-Field and GOLPE Variable Selection Methods in a Study of Inhibitors of Glycogen Phosphorylase b

Cruciani, Gabriele, Watson, Kimberly A.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 3.35 MB

english, 1994

9

Structure-Based Design of HIV-1 Protease Inhibitors: Replacement of Two Amides and a 10.pi.-Aromatic System by a Fused Bis-tetrahydrofuran

Ghosh, Arun K., Thompson, Wayne J., Fitzgerald, Paula M. D., Culberson, J. Chris, Axel, Melinda G., McKee, Sean P., Huff, Joel R., Anderson, Paul S.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.03 MB

english, 1994

10

Synthesis of Naphthalenesulfonic Acid Small Molecules as Selective Inhibitors of the DNA Polymerase and Ribonuclease H Activities of HIV-1 Reverse Transcriptase

Mohan, Prem, Loya, Shoshana, Avidan, Orna, Verma, Sandeep, Dhindsa, Gurnam S., Wong, Man Fai, Huang, Peggy P., Yashiro, Makoto, Baba, Masanori, Hizi, Amnon

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 800 KB

english, 1994

11

Synthesis and Atypical Antipsychotic Profile of Some 2-(2-Piperidinoethyl)benzocycloalkanones as Analogs of Butyrophenone

Fontenla, Jose A., Osuna, Javier, Rosa, Elizabeth, Castro, Ma Elena, G-Ferreiro, Tomas, Loza-Garcia, Isabel, Calleja, Jose M., Sanz, Ferran, Rodriguez, Jesus

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.73 MB

english, 1994

12

GABAA Receptor Agonists, Partial Agonists, and Antagonists. Design and Therapeutic Prospects

Krogsgaard-Larsen, Povl, Froelund, Bente, Joergensen, Flemming S., Schousboe, Arne

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 3.30 MB

english, 1994

13

Maleimidoethyl 3-(Tri-n-butylstannyl)hippurate: A Useful Radioiodination Reagent for Protein Radiopharmaceuticals To Enhance Target Selective Radioactivity Localization

Arano, Yasushi, Wakisaka, Kouji, Ohmomo, Yoshiro, Uezono, Takashi, Mukai, Takahiro, Motonari, Hiroshi, Shiono, Hiromitsu, Sakahara, Harumi, Konishi, Junji

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.83 MB

english, 1994

14

Genetically Evolved Receptor Models: A Computational Approach to Construction of Receptor Models

Walters, D. Eric, Hinds, R. Michael

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.70 MB

english, 1994

15

Synthesis and Structure-Activity Relationships of New Antitumor Taxoids. Effects of Cyclohexyl Substitution at the C-3' and/or C-2 of Taxotere (Docetaxel)

Ojima, Iwao, Duclos, Olivier, Zucco, Martine, Bissery, Marie-Christine, Combeau, C., Vrignaud, P., Riou, J. F., Lavelle, Francois

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.46 MB

english, 1994

16

Synthesis and Biological Properties of5-o-Carboranyl-1-(2-deoxy-2-fluoro-.beta.-D-arabinofuranosyl)uracil

Fulcrand-El Kattan, Geraldine, Goudgaon, Naganna M., Ilksoy, Nurcan, Huang, Jay-Tung, Watanabe, Kyoichi A., Sommadossi, Jean-Pierre, Schinazi, Raymond F.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 775 KB

english, 1994