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Volume 28; Issue 5

Journal of Medicinal Chemistry

Volume 28; Issue 5

1

Synthesis and Antiviral Activity of the Carbocyclic Analogues of (E)-5-(2-Halovinyl)-2'-deoxyuridines and (E)-5-(2-Halovinyl)-2'-deoxycytidines

Herdewijn, Piet, Clercq, Erik De, Balzarini, Jan, Vanderhaeghe, Hubert

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 915 KB

english, 1985

2

Book Reviews

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 162 KB

english, 1985

3

Effect of Structural Modification of the Hydantoin Ring on Anticonvulsant Activity

Cortes, Sergio, Liao, Zeng-Kun, Watson, Darrell, Kohn, Harold

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 789 KB

english, 1985

4

Studies on 4(1H)-Quinazolinones. 5. Synthesis and Antiinflammatory Activity of 4(1H)-Quinazolinone Derivatives

Ozaki, Ken-ichi, Yamada, Yoshihisa, Oine, Toyonari, Ishizuka, Tōru, Iwasawa, Yoshio

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 1.11 MB

english, 1985

5

Studies on Antianaphylactic Agents. 7. Synthesis of Antiallergic 5-Oxo-5H-[1]benzopyrano[2,3-b]pyridines

Nohara, Akira, Ishiguro, Toshihiro, Ukawa, Kiyoshi, Sugihara, Hirosada, Maki, Yoshitaka, Sanno, Yasushi

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 1.28 MB

english, 1985

6

Conjugates of Catecholamines. 5. Synthesis and β-Adrenergic Activity of N-(Aminoalkyl)norepinephrine Derivatives

Reitz, Allen B., Sonveaux, Etienne, Rosenkranz, Roberto P., Verlander, Michael S., Melmon, Kenneth L., Hoffman, Brian B., Akita, Yasio, Castagnoli, Neal, Goodman, Murray

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 1.15 MB

english, 1985

7

Synthesis and Interaction of 5-(Substituted-phenyl)-3-methy1-6,7-dihydropyrazolo[4,3-e][1,4]diazepin-8(7H)-ones with Benzodiazepine Receptors in Rat Cerebral Cortex

Baraldi, Pier Giovanni, Manfredini, Stefano, Periotto, Vittorio, Simoni, Daniele, Guarneri, Mario, Borea, Pier Andrea

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 454 KB

english, 1985

8

New Antihistaminic Theophylline or Theobromine Derivatives

Pascal, Jean-Claude, Beranger, Serge, Pinhas, Henri, Poizot, Alain, Désiles, Jean-Pierre

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 765 KB

english, 1985

9

Methotrexate Analogues. 25. Chemical and Biological Studies on the γ-tert-Butyl Esters of Methotrexate and Aminopterin

Rosowsky, Andre, Freisheim, James H., Bader, Henry, Forsch, Ronald A., Susten, Sandra S., Cucchi, Carol A., Frie, Emil

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 1.26 MB

english, 1985

10

Ibotenic Acid Analogues. Synthesis, Molecular Flexibility, and in Vitro Activity of Agonists and Antagonists at Central Glutamic Acid Receptors

Lauridsen, Jørn, Honoré, Tage, Krogsgaard-Larsen, Povl

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 700 KB

english, 1985

11

Resolution of 5,6-Dihydroxy-2-(N,N-di -n-propylamino)tetralin in Relation to the Structural and Stereochemical Requirements for Centrally Acting Dopamine Agonists

Grol, Cor J., Jansen, Liesbeth J., Rollema, Hans

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 698 KB

english, 1985

12

A New Generation of Phosphodiesterase Inhibitors: Multiple Molecular Forms of Phosphodiesterase and the Potential for Drug Selectivity

Weishaar, Ronald E., Cain, Michael H., Bristol, James A.

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 1.14 MB

english, 1985

13

Quantitative Structure-Activity Relationships in Cytokinin Agonistic and Antagonistic Pyrido[2,3-d]pyrimidine Derivates: Insights into Receptor Topology

Iwamura, Hajime, Murakami, Shigeru, Koshimizu, Koichi, Matsubara, Satoshi

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 910 KB

english, 1985

14

Interactions of Apomorphine with Serum and Tissue Proteins

Smith, Robert V., Velagapudi, Raja B., McLean, Angus M., Wilcox, Richard E.

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 1.21 MB

english, 1985

15

3-Alkyl-3-hydroxyglutaric Acids: A New Class of Hypocholesterolemic HMG CoA Reductase Inhibitors. 1

Baran, John S., Laos, Ivar, Langford, Donna D., Miller, James E., Jett, Charlene, Taite, Beatrice, Rohrbacher, Elaine

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 721 KB

english, 1985

16

Synthesis and Central Dopaminergic Effects of N-(4,6-Dimethyl-2-pyridinyl)benzamides

Bouhayat, Saïd, Piessard, Sylvie, Baut, Guillaume Le, Sparfel, Louis, Petit, Jean-Yves, Piriou, François, Welin, Lucien

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 728 KB

english, 1985

17

Chemistry and Biotechnology of Biologically Active Natural Products. Edited by Cs. Szántay, Á. Gottsegen, and G. Kovács

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 162 KB

english, 1985

18

Masthead

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 153 KB

english, 1985

19

Orally Active and Potent Inhibitors of γ-Aminobutyric Acid Uptake

Ali, Fadia E., Bondinell, William E., Dandridge, Penelope A., Frazee, James S., Garvey, Eleanor, Girard, Gerald R., Kaiser, Carl, Ku, Thomas W., Lafferty, John J., Moonsammy, George I., Oh, Hye-Ja, Ru

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 1.26 MB

english, 1985

20

Phosphorus-Nitrogen Compounds. 26. Phosphaminimides. 2. 2,2'-Phosphinylidenebis(1,1,1-trimethylhydrazinium) Iodide Inner Salts as Agents Affecting Ganglionic Transmission

Cates, Lindley A., Li, Ven-Shun, Saddawi, Bashir H., Alkadhi, Karim A.

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 443 KB

english, 1985

21

1-[3-(Diarylamino)propyl]piperidines and Related Compounds, Potential Antipsychotic Agents with Low Cataleptogenic Profiles

Wise, Lawrence D., Pattison, Ian C., Butler, Donald E., DeWald, Horace A., Lewis, Edward P., Lobbestael, Sandra J., Nordin, Ivan C., Poschel, B. P. H., Coughenour, Linda L.

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 842 KB

english, 1985

22

Conjugates of Catecholamines. 6. Synthesis and β-Adrenergic Activity of N - (Hydroxyalkyl)catecholamine Derivatives

Reitz, Allen B., Avery, Mitchell A., Rosenkranz, Roberto P., Verlander, Michael S., Melmon, Kenneth L., Hoffman, Brian B., Akita, Yasio, Castagnoli, Neal, Goodman, Murry

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 845 KB

english, 1985

23

Aldosterone Antagonists. 1. Synthesis and Activities of 6β,7β:15β,16β-Dimethylene Steroidal Spirolactones

Nickisch, Klaus, Bittler, Dieter, Casals-stenzel, Jorge, Laurent, Henry, Nickolson, Robert, Nishino, Yukishige, Petzoldt, Karl, Wiechert, Rudolf

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 675 KB

english, 1985

24

Synthesis and Structure-Activity Studies on Excitatory Amino Acids Structurally Related to Ibotenic Acid

Krogsgaard-Larsen, Povl, Brehm, Lotte, Johansen, Jørgen S., Vinzents, Peter, Lauridsen, Jørn, Curtis, David R.

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 1000 KB

english, 1985

25

One-Electron Oxidation of Vindoline and 16-O-Acetylvindoline Catalyzed by Peroxidase

Sariaslani, F. Sima, Duffel, M. W., Rosazza, J. P.

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 713 KB

english, 1985

26

"Reverse" and "Symmetrical" Analogues of Actinomycin D: Matabolic Actication and in Vitro and in Vivo Tumor Growth Inhibitory Activities

Sengupta, Sisir K., Kelly, Christinne, Sehgal, Raj K.

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 1.33 MB

english, 1985

27

[(Aminomethy)aryloxy]acetic Acid Esters. A New Class of High-Ceiling Diuretics. 4. Substituted 6,7-Dichloro-2,3-dihydrobenzofurans Derived by Ring Annelation

Lee, Cheuk-Man, Parks, James A., Bunnell, Paul R., Plattner, Jacob J., Field, Michael J., Giebisch, Gerhard H.

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 735 KB

english, 1985

28

Azides and Nitrenes. Reactivity and Utility. Edited by Eric F. V. Scriven

Scheinman, Feodor

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 162 KB

english, 1985

29

Cyclic Melanotropins. 9. 7-D-Phenylalanine Analogues of the Active-Site Sequence

Cody, Wayne L., Mahoney, Mark, Knittel, James J., Hruby, Victor J., Castrucci, Ana Maria de L., Hadley, Mac E.

Journal:

Journal of Medicinal Chemistry

Année:

1985

Langue:

english

Fichier:

PDF, 834 KB

english, 1985