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Stereochemical differences in fluorocyclopropyl amides enable tuning of Btk inhibition and off-target activity
Crawford, James J., Lee, Wendy, Johnson, Adam R., Delatorre, Kelly J, Chen, Jacob, Eigenbrot, Charles, Heidmann, Julia, Kakiuchi-Kiyota, Satoko, Katewa, Arna, Kiefer, James R., Liu, Lichuan, Lubach, JJournal:
ACS Medicinal Chemistry Letters
DOI:
10.1021/acsmedchemlett.0c00249
Date:
July, 2020
Fichier:
PDF, 779 KB
2020