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Discovery of a novel 3,4-dimethylcinnoline carboxamide M4 positive allosteric modulator (PAM) chemotype via scaffold hopping
Temple, Kayla J., Engers, Julie L., Long, Madeline F., Gregro, Alison R., Watson, Katherine J., Chang, Sichen, Jenkins, Matthew T., Luscombe, Vincent B., Rodriguez, Alice L., Niswender, Colleen M., BrLangue:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2019.126678
Date:
September, 2019
Fichier:
PDF, 385 KB
english, 2019