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Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino)cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl)tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor
Wang, Beilei, Wu, Jiaxin, Wu, Yun, Chen, Cheng, Zou, Fengming, Wang, Aoli, Wu, Hong, Hu, Zhenquan, Jiang, Zongru, Liu, Qingwang, Wang, Wei, Zhang, Yicong, Liu, Feiyang, Zhao, Ming, Hu, Jie, Huang, TaoLangue:
english
Journal:
European Journal of Medicinal Chemistry
DOI:
10.1016/j.ejmech.2018.09.025
Date:
September, 2018
Fichier:
PDF, 4.00 MB
english, 2018