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Discovery of ( S )-2-amino- N -(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3Kδ) inhibitor
Liang, Xiaofei, Li, Feng, Chen, Cheng, Jiang, Zongru, Wang, Aoli, Liu, Xiaochuan, Ge, Juan, Hu, Zhenquan, Yu, Kailin, Wang, Wenliang, Zou, Fengming, Liu, Qingwang, Wang, Beilei, Wang, Li, Zhang, ShancVolume:
156
Langue:
english
Journal:
European Journal of Medicinal Chemistry
DOI:
10.1016/j.ejmech.2018.07.036
Date:
August, 2018
Fichier:
PDF, 3.03 MB
english, 2018