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P-glycoprotein (MDR1/ABCB1) restricts brain accumulation and Cytochrome P450-3A (CYP3A) limits oral availability of the novel ALK/ROS1 inhibitor lorlatinib
Li, Wenlong, Sparidans, Rolf W., Wang, Yaogeng, Lebre, Maria C., Wagenaar, Els, Beijnen, Jos H., Schinkel, Alfred H.Langue:
english
Journal:
International Journal of Cancer
DOI:
10.1002/ijc.31582
Date:
May, 2018
Fichier:
PDF, 1.12 MB
english, 2018