Discovery of Novel, Highly Potent, and Selective Matrix Metalloproteinase (MMP)-13 Inhibitors with a 1,2,4-Triazol-3-yl Moiety as a Zinc Binding Group Using a Structure-Based Design Approach
Nara, Hiroshi, Kaieda, Akira, Sato, Kenjiro, Naito, Takako, Mototani, Hideyuki, Oki, Hideyuki, Yamamoto, Yoshio, Kuno, Haruhiko, Santou, Takashi, Kanzaki, Naoyuki, Terauchi, Jun, Uchikawa, Osamu, KoriVolume:
60
Langue:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.6b01007
Date:
January, 2017
Fichier:
PDF, 1.06 MB
english, 2017