Structure-based optimization leads to the discovery of NSC765844, a highly potent, less toxic and orally efficacious dual PI3K/mTOR inhibitor
Han, Jinsong, Chen, Ying, Yang, Chao, Liu, Ting, Wang, Mingping, Xu, Haojie, Zhang, Ling, Zheng, Canhui, Song, Yunlong, Zhu, JuLangue:
english
Journal:
European Journal of Medicinal Chemistry
DOI:
10.1016/j.ejmech.2016.06.030
Date:
June, 2016
Fichier:
PDF, 1.73 MB
english, 2016