Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization and Biological Evaluation
Xue, Xiaoqian, Zhang, Yan, Liu, Zhaoxuan, Song, Ming, Xing, Yanli, Xiang, Qiuping, Wang, Zhen, Tu, Zheng-Chao, Zhou, Yulai, Ding, Ke, Xu, YongLangue:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.5b01511
Date:
January, 2016
Fichier:
PDF, 1.72 MB
english, 2016