Triphenylethanamine Derivatives as Cholesteryl Ester Transfer Protein Inhibitors: Discovery of N -[(1 R )-1-(3-Cyclopropoxy-4-fluorophenyl)-1-[3-fluoro-5-(1,1,2,2-tetrafluoroethoxy)phenyl]-2-phenylethyl]-4-fluoro-3-(trifluoromethyl)benzamide (BMS-795311)
Qiao, Jennifer X., Wang, Tammy C., Adam, Leonard P., Chen, Alice Ye A., Taylor, David S., Yang, Richard Z., Zhuang, Shaobin, Sleph, Paul G., Li, Julia P., Li, Danshi, Yin, Xiaohong, Chang, Ming, Chen,Langue:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.5b01363
Date:
November, 2015
Fichier:
PDF, 1.51 MB
english, 2015