A new structural alert for benzimidazoles: 2,6-Dimethylphenyl substituents increase mutagenic potential and time-dependent CYP3A4 inhibition risk
Youngshin Kwak, Gary Coppola, Cornelia J. Forster, Thomas A. Gilmore, Yongjin Gong, Aaron Kanter, Alan Neubert, Bryan Stroup, Paul Szklennik, Susanne Glowienke, Pascal Stadelmann, Leslie Bell, Shari BVolume:
21
Année:
2011
Langue:
english
Pages:
3
DOI:
10.1016/j.bmcl.2011.01.023
Fichier:
PDF, 382 KB
english, 2011