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Role of Hydrophobic Substituents on the Terminal Nitrogen of Histamine in Receptor Binding and Agonist Activity: Development of an Orally Active Histamine Type 3 Receptor Agonist and Evaluation of Its Antistress Activity in Mice
Ishikawa, Makoto, Shinei, Rie, Yokoyama, Fumikazu, Yamauchi, Miki, Oyama, Masayo, Okuma, Kunihiro, Nagayama, Takako, Kato, Kazuhiko, Kakui, Nobukazu, Sato, YasuoVolume:
53
Langue:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm901890s
Date:
May, 2010
Fichier:
PDF, 837 KB
english, 2010