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Exploiting Protein Fluctuations at the Active-Site Gorge of Human Cholinesterases: Further Optimization of the Design Strategy to Develop Extremely Potent Inhibitors
Butini, Stefania, Campiani, Giuseppe, Borriello, Marianna, Gemma, Sandra, Panico, Alessandro, Persico, Marco, Catalanotti, Bruno, Ros, Sindu, Brindisi, Margherita, Agnusdei, Marianna, Fiorini, IsabellVolume:
51
Langue:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/jm701253t
Date:
June, 2008
Fichier:
PDF, 2.15 MB
english, 2008