Diane H Boschelli : rechercher sur Z-Library

Campagne de collecte 15 septembre 2024 – 1 octobre 2024 C'est quoi, la collecte de fonds?

Le plus grand référentiel d'articles scientifiques au monde. 70,000,000+ d'articles gratuitement.

Campagne de collecte 15 septembre 2024 – 1 octobre 2024

Z-Library est une des plus grandes bibliothèques en ligne dans le monde, avec le stockage de plus de 17,000,000 livres et plus de 84,837,000 articles. Nous encourageons l'accès libre de chacun à la littérature. Aujourd'hui (15 septembre 2024) nous faisons un appel de fonds à tous ceux qui veulent contribuer encore plus au soutien et au développement de notre projet.

Les téléchargements SANS LIMITE sont aussi (au cours de 31 jours après la date de don) disponibles pour TOUS les utilisateurs qui soient en mesure de soutenir le projet pendant la période de collecte de fonds jusqu'au 1 octobre 2024.

C'est quoi, la collecte de fonds?En savoir plus

Livres
Articles (81)
Les plus populaires
Liste
- Liste
- Tableau

51

Further studies on ethenyl and ethynyl-4-phenylamino-3-quinolinecarbonitriles: identification of a subnanomolar Src kinase inhibitor

Ana Carolina Barrios Sosa, Diane H. Boschelli, Biqi Wu, Yan Wang, Jennifer M. Golas

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2005

Langue:

english

Fichier:

PDF, 120 KB

english, 2005

52

A facile, scalable preparation of 4-oxo-4,7-dihydrothieno[2,3-b]pyridine-5-carbonitriles

L. Nathan Tumey, Niala Bhagirath, Biqi Wu, Diane H. Boschelli

Journal:

Tetrahedron Letters

Année:

2008

Langue:

english

Fichier:

PDF, 161 KB

english, 2008

53

ChemInform Abstract: Optimization of 7-Alkene-3-quinolinecarbonitriles as Src Kinase Inhibitors.

Diane H. Boschelli, Daniel Wang, Yan Wang, Biqi Wu, Erick E. Honores, Ana Carolina Barrios Sosa, Inder Chaudhary, Jennifer Golas, Judy Lucas, Frank Boschelli

Journal:

Année:

2010

Fichier:

PDF, 20 KB

2010

54

2-Substituted Aminopyrido[2,3-d]pyrimidin-7(8H)-ones. Structure−Activity Relationships Against Selected Tyrosine Kinases and in Vitro and in Vivo Anticancer Activity

Klutchko, Sylvester R., Hamby, James M., Boschelli, Diane H., Wu, Zhipei, Kraker, Alan J., Amar, Aneesa M., Hartl, Brian G., Shen, Cynthia, Klohs, Wayne D., Steinkampf, Randall W.

Journal:

Journal of Medicinal Chemistry

Année:

1998

Langue:

english

Fichier:

PDF, 404 KB

english, 1998

55

Optimization of 4-Phenylamino-3-quinolinecarbonitriles as Potent Inhibitors of Src Kinase Activity

Boschelli, Diane H., Ye, Fei, Wang, Yanong D., Dutia, Minu, Johnson, Steve L., Wu, Biqi, Miller, Karen, Powell, Dennis W., Yaczko, Deanna, Young, Mairead

Journal:

Journal of Medicinal Chemistry

Année:

2001

Langue:

english

Fichier:

PDF, 245 KB

english, 2001

56

Synthesis and Tyrosine Kinase Inhibitory Activity of a Series of 2-Amino-8H-pyrido[2,3-d]pyrimidines: Identification of Potent, Selective Platelet-Derived Growth Factor Receptor Tyrosine Kinase Inhibitors

Boschelli, Diane H., Wu, Zhipei, Klutchko, Sylvester R., Showalter, H. D. Hollis, Hamby, James M., Lu, Gina H., Major, Terry C., Dahring, Tawny K., Batley, Brian, Panek, Robert L.

Journal:

Journal of Medicinal Chemistry

Année:

1998

Langue:

english

Fichier:

PDF, 219 KB

english, 1998

57

Preparation of Benzothieno[2,3-f]-1,4-oxazepin- and -thiazepin-5(2H)-ones and of Benzothieno[3,2-e]-1,4-diazepin-5-ones

Khatana, Sonya S., Boschelli, Diane H., Kramer, James B., Connor, David T., Barth, Hubert, Stoss, Peter

Journal:

Journal of Organic Chemistry

Année:

1996

Langue:

english

Fichier:

PDF, 156 KB

english, 1996

58

Synthesis and biological properties of 5,10-dideaza-5,6,7,8-tetrahydrofolic acid

Diane H. Boschelli, Stephanie Webber, John M. Whiteley, Arnold L. Oronsky, S.S. Kerwar

Journal:

Archives of Biochemistry and Biophysics

Année:

1988

Langue:

english

Fichier:

PDF, 554 KB

english, 1988

59

Structure−Activity Relationships for 1-Phenylbenzimidazoles as Selective ATP Site Inhibitors of the Platelet-Derived Growth Factor Receptor

Palmer, Brian D., Smaill, Jeff B., Boyd, Maruta, Boschelli, Diane H., Doherty, Annette M., Hamby, James M., Khatana, Sonya S., Kramer, James B., Kraker, Alan J., Panek, Robert L., Lu, Gina H., Dahring

Journal:

Journal of Medicinal Chemistry

Année:

1998

Langue:

english

Fichier:

PDF, 169 KB

english, 1998

60

Synthesis and Src Kinase Inhibitory Activity of 2-Phenyl- and 2-Thienyl-7-phenylaminothieno[3,2- b ]pyridine-6-carbonitriles

Boschelli, Diane H., Wu, Biqi, Barrios Sosa, Ana Carolina, Durutlic, Haris, Chen, Joan J., Wang, Yan, Golas, Jennifer M., Lucas, Judy, Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 197 KB

english, 2005

61

Pyrido[2,3- d ]pyrimidin-7-one Inhi-bitors of Cyclin-Dependent Kinases.

Barvian, Mark, Boschelli, Diane H., Cossrow, Jennifer, Dobrusin, Ellen, Fattaey, Ali, Fritsch, Alex, Fry, David, Harvey, Patricia, Keller, Paul, Garrett, Michelle, La, Frances, Leopold, Wilbur, McNama

Journal:

Journal of Medicinal Chemistry

Année:

2001

Langue:

english

Fichier:

PDF, 15 KB

english, 2001

62

4-Anilino-6,7-dialkoxyquinoline-3-carbonitrile Inhibitors of Epidermal Growth Factor Receptor Kinase and Their Bioisosteric Relationship to the 4-Anilino-6,7-dialkoxyquinazoline Inhibitors

Wissner, Allan, Berger, Dan M., Boschelli, Diane H., Floyd, M. Brawner, Greenberger, Lee M., Gruber, Brian C., Johnson, Bernard D., Mamuya, Nellie, Nilakantan, Ramaswamy, Reich, Marvin F., Shen, Ru, T

Journal:

Journal of Medicinal Chemistry

Année:

2000

Langue:

english

Fichier:

PDF, 384 KB

english, 2000

63

1,3,4-Oxadiazole, 1,3,4-thiadiazole, and 1,2,4-triazole analogs of the fenamates: in vitro inhibition of cyclooxygenase and 5-lipoxygenase activities

Boschelli, Diane H., Connor, David T., Bornemeier, Dirk A., Dyer, Richard D., Kennedy, John A., Kuipers, Paul J., Okonkwo, Godwin C., Schrier, Denis J., Wright, Clifford D.

Journal:

Journal of Medicinal Chemistry

Année:

1993

Langue:

english

Fichier:

PDF, 1.07 MB

english, 1993

64

Identification of 7-Phenylaminothieno- [3,2- b ]pyridine-6-carbonitriles as a New Class of Src Kinase Inhibitors

Boschelli, Diane H., Wu, Biqi, Barrios Sosa, Ana Carolina, Durutlic, Haris, Ye, Fei, Raifeld, Yuri, Golas, Jennifer M., Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Année:

2004

Langue:

english

Fichier:

PDF, 182 KB

english, 2004

65

Discovery of Dibenzo[ c , f ][2,7]naphthyridines as Potent and Selective 3-Phosphoinositide-Dependent Kinase-1 Inhibitors

Gopalsamy, Ariamala, Shi, Mengxiao, Boschelli, Diane H., Williamson, Robert, Olland, Andrea, Hu, Yongbo, Krishnamurthy, Girija, Han, Xin, Arndt, Kim, Guo, Bing

Journal:

Journal of Medicinal Chemistry

Année:

2007

Langue:

english

Fichier:

PDF, 170 KB

english, 2007

66

Pyrido[2,3- d ]pyrimidin-7-one Inhibitors of Cyclin-Dependent Kinases

Barvian, Mark, Boschelli, Diane H., Cossrow, Jennifer, Dobrusin, Ellen, Fattaey, Ali, Fritsch, Alex, Fry, David, Harvey, Patricia, Keller, Paul, Garrett, Michelle, La, Frances, Leopold, Wilbur, McNama

Journal:

Journal of Medicinal Chemistry

Année:

2000

Langue:

english

Fichier:

PDF, 228 KB

english, 2000

67

Inhibition of E-Selectin-, ICAM-1-, and VCAM-1-Mediated Cell Adhesion by Benzo[b]thiophene-, Benzofuran-, Indole-, and Naphthalene-2-carboxamides: Identification of PD 144795 as an Antiinflammatory Agent

Boschelli, Diane H., Kramer, James B., Khatana, Sonya S., Sorenson, Roderick J., Connor, David T., Ferin, Mark A., Wright, Clifford D., Lesch, Mark E., Imre, Kathleen

Journal:

Journal of Medicinal Chemistry

Année:

1995

Langue:

english

Fichier:

PDF, 2.55 MB

english, 1995

68

7-Alkoxy-4-phenylamino-3-quinolinecar-bonitriles as Dual Inhibitors of Src and Abl Kinases

Boschelli, Diane H., Wang, Yanong D., Johnson, Steve, Wu, Biqi, Ye, Fei, Barrios Sosa, Ana Carolina, Golas, Jennifer M., Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Année:

2004

Langue:

english

Fichier:

PDF, 53 KB

english, 2004

69

Benzylidene-thiolactone rearrangement: synthesis and rearrangement of 5-substituted-3-benzylidene-4-thiolen-2-ones

Heindel, Ned D., Conley, Richard A., Minatelli, John A., Boschelli, Diane Harris

Journal:

Journal of Organic Chemistry

Année:

1983

Langue:

english

Fichier:

PDF, 390 KB

english, 1983

70

3-Alkoxybenzo[b]thiophene-2-carboxamides as Inhibitors of Neutrophil-Endothelial Cell Adhesion

Boschelli, Diane H., Kramer, James B., Connor, David T., Lesch, Mark E., Schrier, Denis J., Ferin, Mark A., Wright, Clifford D.

Journal:

Journal of Medicinal Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 256 KB

english, 1994

71

Synthesis and Src Kinase Inhibitory Activity of a Series of 4-[(2,4-Dichloro-5-methoxyphenyl)amino]-7-furyl-3-quinolinecarbonitriles

Boschelli, Diane H., Wu, Biqi, Ye, Fei, Wang, Yan, Golas, Jennifer M., Lucas, Judy, Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 142 KB

english, 2006

72

Stereocontrolled total synthesis of (.+-.)-xanthocidin, two diastereomers, (.+-.)-epixanthocidin and (.+-.)-.beta.-isoxanthocidin, and (.+-.)-dedihydroxy-4,5-didehydroxanthocidin, a likely biosynthetic precursor

Smith, Amos B., Boschelli, Diane

Journal:

Journal of Organic Chemistry

Année:

1983

Langue:

english

Fichier:

PDF, 1.42 MB

english, 1983

73

Synthesis and Src Kinase Inhibitory Activity of a Series of 4-Phenylamino-3-quinolinecarbonitriles

Boschelli, Diane H., Wang, Yanong D., Ye, Fei, Wu, Biqi, Zhang, Nan, Dutia, Minu, Powell, Dennis W., Wissner, Allan, Arndt, Kim, Weber, Jennifer M., Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Année:

2001

Langue:

english

Fichier:

PDF, 162 KB

english, 2001

74

4-Anilino-7,8-dialkoxybenzo[ g ]quinoline-3-carbonitriles as Potent Src Kinase Inhibitors

Berger, Dan M., Dutia, Minu, Birnberg, Gary, Powell, Dennis, Boschelli, Diane H., Wang, Yanong D., Ravi, Malini, Yaczko, Deanna, Golas, Jennifer, Lucas, Judy, Boschelli, Frank

Journal:

Journal of Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 576 KB

english, 2005

75

4-Anilino-3-quinolinecarbonitriles: An Emerging Class of Kinase Inhibitors - An Update

Boschelli, Diane

Journal:

Medicinal Chemistry Reviews - Online

Année:

2004

Langue:

english

Fichier:

PDF, 51 KB

english, 2004

76

4-Anilino-3-quinolinecarbonitriles: An Emerging Class of Kinase Inhibitors

Boschelli, Diane

Journal:

Current Topics in Medicinal Chemistry

Année:

2002

Langue:

english

Fichier:

PDF, 269 KB

english, 2002

77

The Stereospecific Cyclization of A Threo α-Benzamide Alcohol to A Cis N-Acyl Aziridine

Boschelli, Diane Harris

Journal:

Synthetic Communications

Année:

1988

Langue:

english

Fichier:

PDF, 314 KB

english, 1988

78

Editorial [ Hot Topic: Novel Medicinal Chemistry Approaches to New Anti-cancer Agents (Guest Editor: Diane H. Boschelli) ]

Boschelli, Diane

Journal:

Current Topics in Medicinal Chemistry

Année:

2008

Langue:

english

Fichier:

PDF, 13 KB

english, 2008

79

Small Molecule Inhibitors of PKCθ as Potential Antiinflammatory Therapeutics

Boschelli, Diane

Journal:

Current Topics in Medicinal Chemistry

Année:

2009

Langue:

english

Fichier:

PDF, 453 KB

english, 2009

80

Exploitation of the 3-Quinolinecarbonitrile Template for Src Tyrosine Kinase Inhibitors

Boschelli, Diane

Journal:

Current Topics in Medicinal Chemistry

Année:

2008

Langue:

english

Fichier:

PDF, 312 KB

english, 2008

81

A cell-based screen for inhibitors of protein folding and degradation

Frank Boschelli, Jennifer M. Golas, Roseann Petersen, Vincent Lau, Lei Chen, Diane Tkach, Qiang Zhao, Dave S. Fruhling, Hao Liu, Chaneun Nam and Kim T. Arndt

Journal:

Cell Stress and Chaperones

Année:

2010

Langue:

english

Fichier:

PDF, 2.99 MB

english, 2010